Inhibitors | Comment | Organism | Structure |
---|---|---|---|
rolipram | PDE4 is specifically inhibited by rolipram; PDE4 is specifically inhibited by rolipram; PDE4 is specifically inhibited by rolipram; PDE4 is specifically inhibited by rolipram | Homo sapiens |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | P27815 | PDE4A | - |
Homo sapiens | Q07343 | PDE4B | - |
Homo sapiens | Q08493 | PDE4C | - |
Homo sapiens | Q08499 | PDE4D | - |
Homo sapiens | Q13946 | PDE7A | - |
Homo sapiens | Q13946 | PDE7A2 | - |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
umbilical artery smooth muscle | - |
Homo sapiens | - |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
3',5'-cAMP + H2O | specific substrate | Homo sapiens | 5'-AMP | - |
? | |
3',5'-cAMP + H2O | PDE4 hydrolyses selectively 3',5'-cAMP with high affinity | Homo sapiens | 5'-AMP | - |
? |
Synonyms | Comment | Organism |
---|---|---|
PDE4 | key enzyme involved in the regulation of the smooth muscle relaxation associated to cAMP | Homo sapiens |
PDE4A | isoform | Homo sapiens |
PDE4B | isoform | Homo sapiens |
PDE4C | isoform | Homo sapiens |
PDE4D | isoform | Homo sapiens |
PDE7 | - |
Homo sapiens |
PDE7A | isoform | Homo sapiens |
PDE7A2 | isoform | Homo sapiens |