Inhibitors | Comment | Organism | Structure |
---|---|---|---|
(7bS,9R,13bR,15R)-7-amino-9-(hydroxymethyl)-10,13-dioxo-2,3,3a,3b,4,5,6,7,7a,7b,9,10,13,13b-tetradecahydro-1H-6,8-methanobenzo[h]imidazo[1,2-a]pyrido[3,2-c][1,5]naphthyridine-15-carbonitrile | inhibits Cdc25B modestly | Homo sapiens | |
(7bS,9R,13bR,15S)-7-amino-15-hydroxy-9-(hydroxymethyl)-2,3,3a,3b,4,5,6,7,7a,7b,9,13b-dodecahydro-1H-6,8-methanobenzo[h]imidazo[1,2-a]pyrido[3,2-c][1,5]naphthyridine-10,13-dione | - |
Homo sapiens | |
([2-bromo-4-(3-oxo-2,3-diphenylpropyl)phenyl](difluoro)methyl)phosphonic acid | - |
Homo sapiens | |
4-isoavenaciolide | potent irreversible inhibitor of VHR; potent irreversible inhibitor of VHR; potent irreversible inhibitor of VHR | Homo sapiens | |
4-methoxy-3-(5-methoxy-1-benzofuran-6-yl)-5-(4-methoxyphenyl)isoxazole | - |
Homo sapiens | |
4-methoxy-3-(5-methoxy-1-benzofuran-6-yl)-5-phenylisoxazole | - |
Homo sapiens | |
5-(2-fluoro-5-((1E)-3-[3-hydroxy-2-(methoxycarbonyl)phenoxy]prop-1-en-1-yl)phenyl)isoxazole-3-carboxylic acid | - |
Homo sapiens | |
dysidiolide | inhibits Cdc25A | Homo sapiens | |
ethyl-3,4-dephostatin | - |
Homo sapiens | |
hexadecanoyl-5-hydroxymethyl tetronic acid | potent irreversible inhibitor of VHR; potent irreversible inhibitor of VHR; potent irreversible inhibitor of VHR | Homo sapiens | |
kanjone | - |
Homo sapiens | |
karanjin | - |
Homo sapiens | |
menadione | inhibits Cdc25B irreversibly | Homo sapiens | |
methyl 2-[4-[(4-[[ethoxy(oxo)acetyl][2-(methoxycarbonyl)phenyl]amino]-3-ethylphenylalanyl)amino]butoxy]-6-hydroxybenzoate | - |
Homo sapiens | |
nocardione A | inhibits Cdc25B | Homo sapiens | |
nocardione B | inhibits Cdc25B | Homo sapiens | |
Sodium vanadate | - |
Homo sapiens | |
stevastelin | inhibits VHR; inhibits VHR; inhibits VHR | Homo sapiens | |
sulfircin | inhibits Cdc25A | Homo sapiens | |
vanadate | - |
Homo sapiens | |
[(4-[(4E)-2-(1H-benzotriazol-1-yl)-2-[4-(methoxycarbonyl)phenyl]-5-phenylpent-4-en-1-yl]phenyl)(difluoro)methyl]phosphonic acid | - |
Homo sapiens |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | - |
- |
- |
Homo sapiens | P30304 | - |
- |
Homo sapiens | P30305 | Cdc25B | - |
Homo sapiens | P30307 | Cdc25C | - |
Synonyms | Comment | Organism |
---|---|---|
Cdc25A | - |
Homo sapiens |
Cdc25B | - |
Homo sapiens |
Cdc25C | - |
Homo sapiens |
protein tyrosine phosphatase | - |
Homo sapiens |
PTP | - |
Homo sapiens |
PTP1B | - |
Homo sapiens |
VHR | - |
Homo sapiens |
IC50 Value | IC50 Value Maximum | Comment | Organism | Inhibitor | Structure |
---|---|---|---|---|---|
0.0562 | - |
- |
Homo sapiens | Sodium vanadate | |
0.0796 | - |
- |
Homo sapiens | 4-methoxy-3-(5-methoxy-1-benzofuran-6-yl)-5-(4-methoxyphenyl)isoxazole | |
0.0804 | - |
- |
Homo sapiens | 4-methoxy-3-(5-methoxy-1-benzofuran-6-yl)-5-phenylisoxazole |