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Literature summary for 3.1.1.8 extracted from

  • Ahmed, M.; Batista, J.; Rocha, T.; Mazzanti, C.M.; Hassan, W.; Morsch, V.M.; Loro, V.L.; Thome, G.; Schetinger, M.R.
    Comparative study of the inhibitory effect of antidepressants on cholinesterase activity in Bungarus sindanus (krait) venom, human serum and rat striatum (2008), J. Enzyme Inhib. Med. Chem., 23, 912-917.
    View publication on PubMed

Inhibitors

Inhibitors Comment Organism Structure
clomipramine competitive inhibition Homo sapiens
ethopropazine specific inhibitor Homo sapiens
imipramine competitive inhibition Homo sapiens
paroxetine mixed-type inhibition Homo sapiens
sertraline mixed-type inhibition Homo sapiens

Localization

Localization Comment Organism GeneOntology No. Textmining
extracellular
-
Homo sapiens
-
-

Organism

Organism UniProt Comment Textmining
Homo sapiens
-
-
-

Source Tissue

Source Tissue Comment Organism Textmining
heart
-
Homo sapiens
-
intestine
-
Homo sapiens
-
kidney
-
Homo sapiens
-
liver
-
Homo sapiens
-
lung
-
Homo sapiens
-
serum
-
Homo sapiens
-

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
acetylthiocholine + H2O detection with 5,5-dithiobis(2-nitrobenzoic acid) Homo sapiens ?
-
?

Synonyms

Synonyms Comment Organism
acyl choline acylhydrolase
-
Homo sapiens
BuChE
-
Homo sapiens
butyrylcholinesterase
-
Homo sapiens
non specific cholinesterase
-
Homo sapiens
pseudo cholinesterase
-
Homo sapiens

Temperature Optimum [°C]

Temperature Optimum [°C] Temperature Optimum Maximum [°C] Comment Organism
25
-
assay at Homo sapiens

pH Optimum

pH Optimum Minimum pH Optimum Maximum Comment Organism
7.5
-
assay at Homo sapiens