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Literature summary for 3.1.1.4 extracted from

  • Kirincich, S.J.; Xiang, J.; Green, N.; Tam, S.; Yang, H.Y.; Shim, J.; Shen, M.W.; Clark, J.D.; McKew, J.C.
    Benzhydrylquinazolinediones: novel cytosolic phospholipase A2alpha inhibitors with improved physicochemical properties (2009), Bioorg. Med. Chem., 17, 4383-4405.
    View publication on PubMed
Search for more literature for 3.1.1.4

Inhibitors

Inhibitors Comment Organism Structure
(2-(4-((3-(diphenylmethyl)-2,4-dioxo-3,4-dihydroquinazolin-1(2H)-yl)methyl)phenyl)-1,3-oxazol-4-yl)acetic acid
-
 synthetic construct
(4-((3-(diphenylmethyl)-2,4-dioxo-3,4-dihydroquinazolin-1(2H)-yl)methyl)phenoxy)acetic acid
-
 synthetic construct
(4-((3-(diphenylmethyl)-2,4-dioxo-3,4-dihydroquinazolin-1(2H)-yl)methyl)phenyl)acetic acid
-
 synthetic construct
(4-((6-bromo-1-(diphenylmethyl)-2,4-dioxo-1,4-dihydroquinazolin-3(2H)-yl)methyl)phenyl)acetic acid
-
 synthetic construct
2-((6-bromo-1-(diphenylmethyl)-2,4-dioxo-1,4-dihydroquinazolin-3(2H)-yl)methyl)cyclopropanecarboxylic acid
-
 synthetic construct
3-(((2E)-4-(7-chloro-3-(diphenylmethyl)-2,4-dioxo-3,4-dihydroquinazolin-1(2H)-yl)but-2-en-1-yl)oxy)benzoic acid
-
 synthetic construct
4-(((2E)-4-(1-(diphenylmethyl)-2,4-dioxo-1,4-dihydroquinazolin-3(2H)-yl)but-2-en-1-yl)oxy)benzoic acid
-
 synthetic construct
4-(((2E)-4-(1-(diphenylmethyl)-6-fluoro-2,4-dioxo-1,4-dihydroquinazolin-3(2H)-yl)but-2-en-1-yl)oxy)benzoic acid
-
 synthetic construct
4-(((2E)-4-(3-(diphenylmethyl)-2,4-dioxo-3,4-dihydroquinazolin-1(2H)-yl)but-2-en-1-yl)oxy)benzoic acid
-
 synthetic construct
4-(((2E)-4-(3-(diphenylmethyl)-2,4-dioxo-7-(1H-1,2,4-triazol-1-yl)-3,4-dihydroquinazolin-1(2H)-yl)but-2-en-1-yl)oxy)benzoic acid
-
 synthetic construct
4-(((2E)-4-(3-(diphenylmethyl)-2,4-dioxo-7-(phenylthio)-3,4-dihydroquinazolin-1(2H)-yl)but-2-en-1-yl)oxy)benzoic acid
-
 synthetic construct
4-(((2E)-4-(3-(diphenylmethyl)-2,4-dioxo-7-phenoxy-3,4-dihydroquinazolin-1(2H)-yl)but-2-en-1-yl)oxy)benzoic acid
-
 synthetic construct
4-(((2E)-4-(3-(diphenylmethyl)-2,4-dioxo-7-thiomorpholin-4-yl-3,4-dihydroquinazolin-1(2H)-yl)but-2-en-1-yl)oxy)benzoic acid
-
 synthetic construct
4-(((2E)-4-(3-(diphenylmethyl)-6-fluoro-2,4-dioxo-3,4-dihydroquinazolin-1(2H)-yl)but-2-en-1-yl)oxy)benzoic acid
-
 synthetic construct
4-(((2E)-4-(3-(diphenylmethyl)-7-(4-(methoxycarbonyl)piperidin-1-yl)-2,4-dioxo-3,4-dihydroquinazolin-1(2H)-yl)but-2-en-1-yl)oxy)benzoic acid
-
 synthetic construct
4-(((2E)-4-(3-(diphenylmethyl)-7-(methylsulfonyl)-2,4-dioxo-3,4-dihydroquinazolin-1(2H)-yl)but-2-en-1-yl)oxy)benzoic acid
-
 synthetic construct
4-(((2E)-4-(3-(diphenylmethyl)-7-(methylthio)-2,4-dioxo-3,4-dihydroquinazolin-1(2H)-yl)but-2-en-1-yl)oxy)benzoic acid
-
 synthetic construct
4-(((2E)-4-(3-(diphenylmethyl)-7-fluoro-2,4-dioxo-3,4-dihydroquinazolin-1(2H)-yl)but-2-en-1-yl)oxy)benzoic acid
-
 synthetic construct
4-(((2E)-4-(3-(diphenylmethyl)-7-methoxy-2,4-dioxo-3,4-dihydroquinazolin-1(2H)-yl)but-2-en-1-yl)oxy)benzoic acid
-
 synthetic construct
4-(((2E)-4-(3-(diphenylmethyl)-7-methyl-2,4-dioxo-3,4-dihydroquinazolin-1(2H)-yl)but-2-en-1-yl)oxy)benzoic acid
-
 synthetic construct
4-(((2E)-4-(3-(diphenylmethyl)-7-morpholin-4-yl-2,4-dioxo-3,4-dihydroquinazolin-1(2H)-yl)but-2-en-1-yl)oxy)benzoic acid
-
 synthetic construct
4-(((2E)-4-(3-(diphenylmethyl)-7-nitro-2,4-dioxo-3,4-dihydroquinazolin-1(2H)-yl)but-2-en-1-yl)oxy)benzoic acid
-
 synthetic construct
4-(((2E)-4-(6-chloro-3-(diphenylmethyl)-2,4-dioxo-3,4-dihydroquinazolin-1(2H)-yl)but-2-en-1-yl)oxy)benzoic acid
-
 synthetic construct
4-(((2E)-4-(7-amino-3-(diphenylmethyl)-2,4-dioxo-3,4-dihydroquinazolin-1(2H)-yl)but-2-en-1-yl)oxy)benzoic acid
-
 synthetic construct
4-(((2E)-4-(7-chloro-1-(diphenylmethyl)-2,4-dioxo-1,4-dihydroquinazolin-3(2H)-yl)but-2-en-1-yl)oxy)benzoic acid
-
 synthetic construct
4-(((2E)-4-(7-chloro-3-(diphenylmethyl)-2,4-dioxo-3,4-dihydroquinazolin-1(2H)-yl)but-2-en-1-yl)oxy)benzoic acid
-
 synthetic construct
4-(((2E)-4-[1-(diphenylmethyl)-2,4-dioxo-1,4-dihydroquinazolin-3(2H)-yl]but-2-en-1-yl)oxy)benzoic acid
-
 Rattus norvegicus
4-(((2E)-4-[3-(diphenylmethyl)-2,4-dioxo-3,4-dihydroquinazolin-1(2H)-yl]but-2-en-1-yl)oxy)benzoic acid
-
 Rattus norvegicus
4-(((2E)-4-[3-(diphenylmethyl)-2,4-dioxo-7-(1H-1,2,4-triazol-1-yl)-3,4-dihydroquinazolin-1(2H)-yl]but-2-en-1-yl)oxy)benzoic acid
-
 Rattus norvegicus
4-(((2E)-4-[3-(diphenylmethyl)-7-fluoro-2,4-dioxo-3,4-dihydroquinazolin-1(2H)-yl]but-2-en-1-yl)oxy)benzoic acid
-
 Rattus norvegicus
4-(((2E)-4-[3-(diphenylmethyl)-7-methoxy-2,4-dioxo-3,4-dihydroquinazolin-1(2H)-yl]but-2-en-1-yl)oxy)benzoic acid
-
 Rattus norvegicus
4-(((2E)-4-[3-(diphenylmethyl)-7-nitro-2,4-dioxo-3,4-dihydroquinazolin-1(2H)-yl]but-2-en-1-yl)oxy)benzoic acid
-
 Rattus norvegicus
4-(((2E)-4-[7-chloro-3-(diphenylmethyl)-2,4-dioxo-3,4-dihydroquinazolin-1(2H)-yl]but-2-en-1-yl)oxy)benzoic acid
-
 Rattus norvegicus
4-(((2Z)-4-(1-(diphenylmethyl)-2,4-dioxo-1,4-dihydroquinazolin-3(2H)-yl)but-2-en-1-yl)oxy)benzoic acid
-
 synthetic construct
4-(((2Z)-4-(3-(diphenylmethyl)-2,4-dioxo-3,4-dihydroquinazolin-1(2H)-yl)but-2-en-1-yl)oxy)benzoic acid
-
 synthetic construct
4-(((2Z)-4-(3-(diphenylmethyl)-6-fluoro-2,4-dioxo-3,4-dihydroquinazolin-1(2H)-yl)but-2-en-1-yl)oxy)benzoic acid
-
 synthetic construct
4-(((2Z)-4-(6-bromo-3-(diphenylmethyl)-2,4-dioxo-3,4-dihydroquinazolin-1(2H)-yl)but-2-en-1-yl)oxy)benzoic acid
-
 synthetic construct
4-(((2Z)-4-(6-chloro-3-(diphenylmethyl)-2,4-dioxo-3,4-dihydroquinazolin-1(2H)-yl)but-2-en-1-yl)oxy)benzoic acid
-
 synthetic construct
4-(((2Z)-4-(7-chloro-1-(diphenylmethyl)-2,4-dioxo-1,4-dihydroquinazolin-3(2H)-yl)but-2-en-1-yl)oxy)benzoic acid
-
 synthetic construct
4-(((2Z)-4-(7-chloro-3-(diphenylmethyl)-2,4-dioxo-3,4-dihydroquinazolin-1(2H)-yl)but-2-en-1-yl)oxy)benzoic acid
-
 synthetic construct
4-(((E)-4-(3-benzhydryl-6-bromo-2,4-dioxo-3,4-dihydro-1(2H)-quinazolinyl)-2-butenyl)oxy)benzoic acid
-
 synthetic construct
4-((5-(3-(diphenylmethyl)-2,4-dioxo-3,4-dihydroquinazolin-1(2H)-yl)pentyl)oxy)benzoic acid
-
 synthetic construct
4-((6-(3-(diphenylmethyl)-2,4-dioxo-3,4-dihydroquinazolin-1(2H)-yl)hexyl)oxy)benzoic acid
-
 synthetic construct
4-((6-chloro-1-(diphenylmethyl)-2,4-dioxo-1,4-dihydroquinazolin-3(2H)-yl)methyl)benzoic acid
-
 synthetic construct
4-((7-(3-(diphenylmethyl)-2,4-dioxo-3,4-dihydroquinazolin-1(2H)-yl)heptyl)oxy)benzoic acid
-
 synthetic construct
4-((7-chloro-1-(diphenylmethyl)-2,4-dioxo-1,4-dihydroquinazolin-3(2H)-yl)methyl)benzoic acid
-
 synthetic construct
4-(2-(1-(diphenylmethyl)-2,4-dioxo-1,4-dihydroquinazolin-3(2H)-yl)ethoxy)benzoic acid
-
 synthetic construct
4-(2-(1-benzyl-2,4-dioxo-1,4-dihydroquinazolin-3(2H)-yl)ethoxy)benzoic acid
-
 synthetic construct
4-(2-(7-chloro-1-(diphenylmethyl)-2,4-dioxo-1,4-dihydroquinazolin-3(2H)-yl)ethoxy)benzoic acid
-
 synthetic construct
4-(2-(7-chloro-3-(diphenylmethyl)-2,4-dioxo-3,4-dihydroquinazolin-1(2H)-yl)ethoxy)benzoic acid
-
 synthetic construct
4-(3-(3-(diphenylmethyl)-2,4-dioxo-3,4-dihydroquinazolin-1(2H)-yl)propoxy)benzoic acid
-
 synthetic construct
4-(4-((3-(diphenylmethyl)-2,4-dioxo-3,4-dihydroquinazolin-1(2H)-yl)methyl)phenoxy)butanoic acid
-
 synthetic construct
4-(4-(7-chloro-3-(diphenylmethyl)-2,4-dioxo-3,4-dihydroquinazolin-1(2H)-yl)butoxy)benzoic acid
-
 synthetic construct

Organism

Organism UniProt Comment Textmining
Rattus norvegicus
-
-
-
synthetic construct
-
-
-

Source Tissue

Source Tissue Comment Organism Textmining
blood
-
 Rattus norvegicus
-

Synonyms

Synonyms Comment Organism
cPLA2alpha
-
 Rattus norvegicus
cPLA2alpha
-
 synthetic construct
cytosolic phospholipase A2alpha
-
 Rattus norvegicus
cytosolic phospholipase A2alpha
-
 synthetic construct

IC50 Value

IC50 Value IC50 Value Maximum Comment Organism Inhibitor Structure
0.001
-
 7-hydroxycoumarinyl-gamma-linoleolate micelle assay synthetic construct 4-(((2E)-4-(7-chloro-3-(diphenylmethyl)-2,4-dioxo-3,4-dihydroquinazolin-1(2H)-yl)but-2-en-1-yl)oxy)benzoic acid
0.001
-
 7-hydroxycoumarinyl-gamma-linoleolate micelle assay synthetic construct 4-(((2E)-4-(3-(diphenylmethyl)-7-nitro-2,4-dioxo-3,4-dihydroquinazolin-1(2H)-yl)but-2-en-1-yl)oxy)benzoic acid
0.0011
-
 7-hydroxycoumarinyl-gamma-linoleolate micelle assay synthetic construct 4-(((2E)-4-(3-(diphenylmethyl)-2,4-dioxo-7-(1H-1,2,4-triazol-1-yl)-3,4-dihydroquinazolin-1(2H)-yl)but-2-en-1-yl)oxy)benzoic acid
0.0014
-
 7-hydroxycoumarinyl-gamma-linoleolate micelle assay synthetic construct 4-(((2E)-4-(3-(diphenylmethyl)-7-fluoro-2,4-dioxo-3,4-dihydroquinazolin-1(2H)-yl)but-2-en-1-yl)oxy)benzoic acid
0.0016
-
 7-hydroxycoumarinyl-gamma-linoleolate micelle assay synthetic construct 4-(((2E)-4-(3-(diphenylmethyl)-2,4-dioxo-7-phenoxy-3,4-dihydroquinazolin-1(2H)-yl)but-2-en-1-yl)oxy)benzoic acid
0.0018
-
 7-hydroxycoumarinyl-gamma-linoleolate micelle assay synthetic construct 4-(((2E)-4-(3-(diphenylmethyl)-7-(4-(methoxycarbonyl)piperidin-1-yl)-2,4-dioxo-3,4-dihydroquinazolin-1(2H)-yl)but-2-en-1-yl)oxy)benzoic acid
0.002
-
 7-hydroxycoumarinyl-gamma-linoleolate micelle assay synthetic construct 4-(((2E)-4-(1-(diphenylmethyl)-2,4-dioxo-1,4-dihydroquinazolin-3(2H)-yl)but-2-en-1-yl)oxy)benzoic acid
0.002
-
 7-hydroxycoumarinyl-gamma-linoleolate micelle assay synthetic construct 4-(((2E)-4-(3-(diphenylmethyl)-7-(methylthio)-2,4-dioxo-3,4-dihydroquinazolin-1(2H)-yl)but-2-en-1-yl)oxy)benzoic acid
0.0021
-
 7-hydroxycoumarinyl-gamma-linoleolate micelle assay synthetic construct 4-(((2E)-4-(3-(diphenylmethyl)-2,4-dioxo-7-(phenylthio)-3,4-dihydroquinazolin-1(2H)-yl)but-2-en-1-yl)oxy)benzoic acid
0.0022
-
 7-hydroxycoumarinyl-gamma-linoleolate micelle assay synthetic construct 4-(((2E)-4-(3-(diphenylmethyl)-7-morpholin-4-yl-2,4-dioxo-3,4-dihydroquinazolin-1(2H)-yl)but-2-en-1-yl)oxy)benzoic acid
0.0024
-
 7-hydroxycoumarinyl-gamma-linoleolate micelle assay synthetic construct 4-(((2E)-4-(3-(diphenylmethyl)-2,4-dioxo-7-thiomorpholin-4-yl-3,4-dihydroquinazolin-1(2H)-yl)but-2-en-1-yl)oxy)benzoic acid
0.0025
-
 7-hydroxycoumarinyl-gamma-linoleolate micelle assay synthetic construct 4-(4-(7-chloro-3-(diphenylmethyl)-2,4-dioxo-3,4-dihydroquinazolin-1(2H)-yl)butoxy)benzoic acid
0.0028
-
 7-hydroxycoumarinyl-gamma-linoleolate micelle assay synthetic construct 4-(((2E)-4-(3-(diphenylmethyl)-7-methyl-2,4-dioxo-3,4-dihydroquinazolin-1(2H)-yl)but-2-en-1-yl)oxy)benzoic acid
0.003
-
 7-hydroxycoumarinyl-gamma-linoleolate micelle assay synthetic construct 4-(((2E)-4-(3-(diphenylmethyl)-2,4-dioxo-3,4-dihydroquinazolin-1(2H)-yl)but-2-en-1-yl)oxy)benzoic acid
0.003
-
 7-hydroxycoumarinyl-gamma-linoleolate micelle assay synthetic construct 4-(((2E)-4-(3-(diphenylmethyl)-7-methoxy-2,4-dioxo-3,4-dihydroquinazolin-1(2H)-yl)but-2-en-1-yl)oxy)benzoic acid
0.004
-
 7-hydroxycoumarinyl-gamma-linoleolate micelle assay synthetic construct 4-(2-(7-chloro-1-(diphenylmethyl)-2,4-dioxo-1,4-dihydroquinazolin-3(2H)-yl)ethoxy)benzoic acid
0.0045
-
 7-hydroxycoumarinyl-gamma-linoleolate micelle assay synthetic construct 4-(((2E)-4-(7-chloro-1-(diphenylmethyl)-2,4-dioxo-1,4-dihydroquinazolin-3(2H)-yl)but-2-en-1-yl)oxy)benzoic acid
0.0056
-
 7-hydroxycoumarinyl-gamma-linoleolate micelle assay synthetic construct 4-(((2E)-4-(1-(diphenylmethyl)-6-fluoro-2,4-dioxo-1,4-dihydroquinazolin-3(2H)-yl)but-2-en-1-yl)oxy)benzoic acid
0.006
-
 whole blood assay Rattus norvegicus 4-(((2E)-4-[3-(diphenylmethyl)-7-fluoro-2,4-dioxo-3,4-dihydroquinazolin-1(2H)-yl]but-2-en-1-yl)oxy)benzoic acid
0.006
-
 7-hydroxycoumarinyl-gamma-linoleolate micelle assay synthetic construct 4-(((2E)-4-(3-(diphenylmethyl)-6-fluoro-2,4-dioxo-3,4-dihydroquinazolin-1(2H)-yl)but-2-en-1-yl)oxy)benzoic acid
0.009
-
 whole blood assay Rattus norvegicus 4-(((2E)-4-[3-(diphenylmethyl)-7-methoxy-2,4-dioxo-3,4-dihydroquinazolin-1(2H)-yl]but-2-en-1-yl)oxy)benzoic acid
0.009
-
 7-hydroxycoumarinyl-gamma-linoleolate micelle assay synthetic construct 4-(((E)-4-(3-benzhydryl-6-bromo-2,4-dioxo-3,4-dihydro-1(2H)-quinazolinyl)-2-butenyl)oxy)benzoic acid
0.009
-
 7-hydroxycoumarinyl-gamma-linoleolate micelle assay synthetic construct 4-(((2E)-4-(7-amino-3-(diphenylmethyl)-2,4-dioxo-3,4-dihydroquinazolin-1(2H)-yl)but-2-en-1-yl)oxy)benzoic acid
0.01
-
 7-hydroxycoumarinyl-gamma-linoleolate micelle assay synthetic construct 4-(2-(1-(diphenylmethyl)-2,4-dioxo-1,4-dihydroquinazolin-3(2H)-yl)ethoxy)benzoic acid
0.01
-
 7-hydroxycoumarinyl-gamma-linoleolate micelle assay synthetic construct 4-(2-(7-chloro-3-(diphenylmethyl)-2,4-dioxo-3,4-dihydroquinazolin-1(2H)-yl)ethoxy)benzoic acid
0.01
-
 7-hydroxycoumarinyl-gamma-linoleolate micelle assay synthetic construct 4-(((2E)-4-(6-chloro-3-(diphenylmethyl)-2,4-dioxo-3,4-dihydroquinazolin-1(2H)-yl)but-2-en-1-yl)oxy)benzoic acid
0.011
-
 whole blood assay Rattus norvegicus 4-(((2E)-4-[7-chloro-3-(diphenylmethyl)-2,4-dioxo-3,4-dihydroquinazolin-1(2H)-yl]but-2-en-1-yl)oxy)benzoic acid
0.011
-
 whole blood assay Rattus norvegicus 4-(((2E)-4-[3-(diphenylmethyl)-2,4-dioxo-7-(1H-1,2,4-triazol-1-yl)-3,4-dihydroquinazolin-1(2H)-yl]but-2-en-1-yl)oxy)benzoic acid
0.012
-
 whole blood assay Rattus norvegicus 4-(((2E)-4-[1-(diphenylmethyl)-2,4-dioxo-1,4-dihydroquinazolin-3(2H)-yl]but-2-en-1-yl)oxy)benzoic acid
0.012
-
 7-hydroxycoumarinyl-gamma-linoleolate micelle assay synthetic construct (4-((6-bromo-1-(diphenylmethyl)-2,4-dioxo-1,4-dihydroquinazolin-3(2H)-yl)methyl)phenyl)acetic acid
0.013
-
 whole blood assay Rattus norvegicus 4-(((2E)-4-[3-(diphenylmethyl)-7-nitro-2,4-dioxo-3,4-dihydroquinazolin-1(2H)-yl]but-2-en-1-yl)oxy)benzoic acid
0.014
-
 whole blood assay Rattus norvegicus 4-(((2E)-4-[3-(diphenylmethyl)-2,4-dioxo-3,4-dihydroquinazolin-1(2H)-yl]but-2-en-1-yl)oxy)benzoic acid
0.015
-
 7-hydroxycoumarinyl-gamma-linoleolate micelle assay synthetic construct 4-(((2E)-4-(3-(diphenylmethyl)-7-(methylsulfonyl)-2,4-dioxo-3,4-dihydroquinazolin-1(2H)-yl)but-2-en-1-yl)oxy)benzoic acid
0.025
-
 7-hydroxycoumarinyl-gamma-linoleolate micelle assay synthetic construct 4-(((2Z)-4-(1-(diphenylmethyl)-2,4-dioxo-1,4-dihydroquinazolin-3(2H)-yl)but-2-en-1-yl)oxy)benzoic acid
0.03
-
 7-hydroxycoumarinyl-gamma-linoleolate micelle assay synthetic construct 4-((5-(3-(diphenylmethyl)-2,4-dioxo-3,4-dihydroquinazolin-1(2H)-yl)pentyl)oxy)benzoic acid
0.03
-
 7-hydroxycoumarinyl-gamma-linoleolate micelle assay synthetic construct 4-(((2Z)-4-(6-bromo-3-(diphenylmethyl)-2,4-dioxo-3,4-dihydroquinazolin-1(2H)-yl)but-2-en-1-yl)oxy)benzoic acid
0.03
-
 7-hydroxycoumarinyl-gamma-linoleolate micelle assay synthetic construct 4-(((2Z)-4-(7-chloro-3-(diphenylmethyl)-2,4-dioxo-3,4-dihydroquinazolin-1(2H)-yl)but-2-en-1-yl)oxy)benzoic acid
0.04
-
 7-hydroxycoumarinyl-gamma-linoleolate micelle assay synthetic construct 4-(4-((3-(diphenylmethyl)-2,4-dioxo-3,4-dihydroquinazolin-1(2H)-yl)methyl)phenoxy)butanoic acid
0.04
-
 7-hydroxycoumarinyl-gamma-linoleolate micelle assay synthetic construct 4-(((2Z)-4-(3-(diphenylmethyl)-6-fluoro-2,4-dioxo-3,4-dihydroquinazolin-1(2H)-yl)but-2-en-1-yl)oxy)benzoic acid
0.04
-
 7-hydroxycoumarinyl-gamma-linoleolate micelle assay synthetic construct 4-(((2Z)-4-(6-chloro-3-(diphenylmethyl)-2,4-dioxo-3,4-dihydroquinazolin-1(2H)-yl)but-2-en-1-yl)oxy)benzoic acid
0.044
-
 7-hydroxycoumarinyl-gamma-linoleolate micelle assay synthetic construct 4-(((2Z)-4-(3-(diphenylmethyl)-2,4-dioxo-3,4-dihydroquinazolin-1(2H)-yl)but-2-en-1-yl)oxy)benzoic acid
0.047
-
 7-hydroxycoumarinyl-gamma-linoleolate micelle assay synthetic construct 4-((6-(3-(diphenylmethyl)-2,4-dioxo-3,4-dihydroquinazolin-1(2H)-yl)hexyl)oxy)benzoic acid
0.05
-
 7-hydroxycoumarinyl-gamma-linoleolate micelle assay synthetic construct 4-(3-(3-(diphenylmethyl)-2,4-dioxo-3,4-dihydroquinazolin-1(2H)-yl)propoxy)benzoic acid
0.06
-
 7-hydroxycoumarinyl-gamma-linoleolate micelle assay synthetic construct 4-(((2Z)-4-(7-chloro-1-(diphenylmethyl)-2,4-dioxo-1,4-dihydroquinazolin-3(2H)-yl)but-2-en-1-yl)oxy)benzoic acid
0.071
-
 7-hydroxycoumarinyl-gamma-linoleolate micelle assay synthetic construct 4-((7-(3-(diphenylmethyl)-2,4-dioxo-3,4-dihydroquinazolin-1(2H)-yl)heptyl)oxy)benzoic acid
0.08
-
 7-hydroxycoumarinyl-gamma-linoleolate micelle assay synthetic construct 4-((7-chloro-1-(diphenylmethyl)-2,4-dioxo-1,4-dihydroquinazolin-3(2H)-yl)methyl)benzoic acid
0.09
-
 7-hydroxycoumarinyl-gamma-linoleolate micelle assay synthetic construct 4-((6-chloro-1-(diphenylmethyl)-2,4-dioxo-1,4-dihydroquinazolin-3(2H)-yl)methyl)benzoic acid
0.1
-
 7-hydroxycoumarinyl-gamma-linoleolate micelle assay synthetic construct 4-(2-(1-benzyl-2,4-dioxo-1,4-dihydroquinazolin-3(2H)-yl)ethoxy)benzoic acid
0.1
-
 7-hydroxycoumarinyl-gamma-linoleolate micelle assay synthetic construct 3-(((2E)-4-(7-chloro-3-(diphenylmethyl)-2,4-dioxo-3,4-dihydroquinazolin-1(2H)-yl)but-2-en-1-yl)oxy)benzoic acid
0.12
-
 7-hydroxycoumarinyl-gamma-linoleolate micelle assay synthetic construct 2-((6-bromo-1-(diphenylmethyl)-2,4-dioxo-1,4-dihydroquinazolin-3(2H)-yl)methyl)cyclopropanecarboxylic acid
0.14
-
 7-hydroxycoumarinyl-gamma-linoleolate micelle assay synthetic construct (2-(4-((3-(diphenylmethyl)-2,4-dioxo-3,4-dihydroquinazolin-1(2H)-yl)methyl)phenyl)-1,3-oxazol-4-yl)acetic acid
0.26
-
 7-hydroxycoumarinyl-gamma-linoleolate micelle assay synthetic construct (4-((3-(diphenylmethyl)-2,4-dioxo-3,4-dihydroquinazolin-1(2H)-yl)methyl)phenyl)acetic acid
0.36
-
 7-hydroxycoumarinyl-gamma-linoleolate micelle assay synthetic construct (4-((3-(diphenylmethyl)-2,4-dioxo-3,4-dihydroquinazolin-1(2H)-yl)methyl)phenoxy)acetic acid