Inhibitors | Comment | Organism | Structure |
---|---|---|---|
2,2-Difluorosuccinate | strong | Rattus norvegicus | |
3-Sulfopropanoate | - |
Rattus norvegicus | |
acetoacetate | - |
Rattus norvegicus | |
acetylene dicarboxylate | weak | Rattus norvegicus | |
Maleamate | reversible, competitive | Rattus norvegicus | |
Maleimide | succinate or acetoacetate protects | Rattus norvegicus | |
malonate | kinetics | Rattus norvegicus | |
Monomethylsuccinate | competitive | Rattus norvegicus | |
additional information | no inhibition by glutarate, adipate, cis- or trans-cyclobutane-1,2-dicarboxylate, cis- or trans-cyclohexane-1,2-dicarboxylate, methylsuccinate, mercaptosuccinate, malate, aspartate, succinimide or iodoacetamide | Rattus norvegicus | |
N-ethylmaleamate | reversible, competitive | Rattus norvegicus | |
N-ethylmaleimide | succinate or acetoacetate protects | Rattus norvegicus | |
oxalate | kinetics | Rattus norvegicus | |
Perfluorosuccinate | strong | Rattus norvegicus | |
succinamate | competitive | Rattus norvegicus | |
succinate | product inhibition | Rattus norvegicus |
KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.04 | - |
acetoacetyl-CoA | pH 8.1, 25°C | Rattus norvegicus | |
0.28 | - |
succinyl-CoA | pH 8.1, 25°C | Rattus norvegicus | |
0.44 | - |
acetoacetate | pH 8.1, 25°C | Rattus norvegicus | |
28 | - |
succinate | cosusbstrate: acetoacetyl-CoA, pH 8.1, 25°C | Rattus norvegicus | |
35 | - |
Maleate | cosusbstrate: acetoacetyl-CoA, pH 8.1, 25°C | Rattus norvegicus |
Localization | Comment | Organism | GeneOntology No. | Textmining |
---|---|---|---|---|
mitochondrion | - |
Rattus norvegicus | 5739 | - |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Rattus norvegicus | - |
male adult Buffalo | - |
Purification (Comment) | Organism |
---|---|
partial | Rattus norvegicus |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
heart | - |
Rattus norvegicus | - |
Specific Activity Minimum [µmol/min/mg] | Specific Activity Maximum [µmol/min/mg] | Comment | Organism |
---|---|---|---|
2.88 | - |
- |
Rattus norvegicus |
Storage Stability | Organism |
---|---|
frozen, partially purified preparation in phosphate solution, less than 10% loss of activity within 1-2 weeks | Rattus norvegicus |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
additional information | no substrates are diacids with connecting chain lengths of 3 or more methylene groups | Rattus norvegicus | ? | - |
? | |
succinyl-CoA + acetoacetate | - |
Rattus norvegicus | succinate + acetoacetyl-CoA | - |
r | |
succinyl-CoA + maleate | - |
Rattus norvegicus | succinate + maleyl-CoA | - |
? |
Temperature Optimum [°C] | Temperature Optimum Maximum [°C] | Comment | Organism |
---|---|---|---|
25 | - |
assay at | Rattus norvegicus |
Ki Value [mM] | Ki Value maximum [mM] | Inhibitor | Comment | Organism | Structure |
---|---|---|---|---|---|
0.72 | - |
succinate | pH 8.1, 25°C | Rattus norvegicus | |
3.7 | - |
acetoacetate | pH 8.1, 25°C | Rattus norvegicus | |
6.4 | - |
2,2-Difluorosuccinate | pH 8.1, 25°C | Rattus norvegicus | |
15 | - |
oxalate | pH 8.1, 25°C | Rattus norvegicus | |
18 | - |
Perfluorosuccinate | pH 8.1, 25°C | Rattus norvegicus | |
21 | - |
malonate | pH 8.1, 25°C | Rattus norvegicus |