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Literature summary for 2.8.2.20 extracted from

  • Danan, L.M.; Yu, Z.; Ludden, P.J.; Jia, W.; Moore, K.L.; Leary, J.A.
    Catalytic mechanism of Golgi-resident human tyrosylprotein sulfotransferase-2: a mass spectrometry approach (2010), J. Am. Soc. Mass Spectrom., 21, 1633-1642.
    View publication on PubMedView publication on EuropePMC

Cloned(Commentary)

Cloned (Comment) Organism
expressed in CHO-K1 cells Homo sapiens

Inhibitors

Inhibitors Comment Organism Structure
adenosine 3',5'-bisphosphate product inhibition Homo sapiens

KM Value [mM]

KM Value [mM] KM Value Maximum [mM] Substrate Comment Organism Structure
0.0031
-
VTDsYYYPDI in 20 mM MOPS, at pH 7.5, 100 mM NaCl, at 30°C Homo sapiens
0.0048
-
3'-phosphoadenylyl sulfate with VTDsYYYPDI as cosubstrate, in 20 mM MOPS, at pH 7.5, 100 mM NaCl, at 30°C Homo sapiens
0.0087
-
3'-phosphoadenylyl sulfate with VTDYYYPDI as cosubstrate, in 20 mM MOPS, at pH 7.5, 100 mM NaCl, at 30°C Homo sapiens
0.0193
-
VTDYYYPDI in 20 mM MOPS, at pH 7.5, 100 mM NaCl, at 30°C Homo sapiens

Localization

Localization Comment Organism GeneOntology No. Textmining
Golgi apparatus
-
Homo sapiens 5794
-

Natural Substrates/ Products (Substrates)

Natural Substrates Organism Comment (Nat. Sub.) Natural Products Comment (Nat. Pro.) Rev. Reac.
3'-phosphoadenylyl sulfate + VTDsYYYPDI Homo sapiens
-
adenosine 3',5'-bisphosphate + VTDsYYsYPDI
-
ir
3'-phosphoadenylyl sulfate + VTDYYYPDI Homo sapiens
-
adenosine 3',5'-bisphosphate + VTDsYYYPDI
-
ir

Organism

Organism UniProt Comment Textmining
Homo sapiens
-
-
-

Purification (Commentary)

Purification (Comment) Organism
HPC4 affinity column chromatography, and gel filtration Homo sapiens

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
3'-phosphoadenylyl sulfate + VTDsYYYPDI
-
Homo sapiens adenosine 3',5'-bisphosphate + VTDsYYsYPDI
-
ir
3'-phosphoadenylyl sulfate + VTDYYYPDI
-
Homo sapiens adenosine 3',5'-bisphosphate + VTDsYYYPDI
-
ir

Synonyms

Synonyms Comment Organism
TPST-2
-
Homo sapiens
tyrosylprotein sulfotransferase-2
-
Homo sapiens

Ki Value [mM]

Ki Value [mM] Ki Value maximum [mM] Inhibitor Comment Organism Structure
0.00016
-
adenosine 3',5'-bisphosphate with VTDsYYYPDI as substrate, in 20 mM MOPS, at pH 7.5, 100 mM NaCl, at 30°C Homo sapiens
0.00074
-
adenosine 3',5'-bisphosphate with VTDYYYPDI as substrate, in 20 mM MOPS, at pH 7.5, 100 mM NaCl, at 30°C Homo sapiens