Protein Variants | Comment | Organism |
---|---|---|
K65R | mutant maintains a susceptibility to GS-9148 that is similar to wild type enzyme | Human immunodeficiency virus 1 |
M184V | mutant maintains a susceptibility to GS-9148 that is similar to wild type enzyme | Human immunodeficiency virus 1 |
Inhibitors | Comment | Organism | Structure |
---|---|---|---|
([[(2R,5R)-5-(6-amino-7H-purin-7-yl)-2,5-dihydrofuran-2-yl]oxy]methyl)phosphonic acid | - |
Human immunodeficiency virus 1 | |
([[(2R,5R)-5-(6-amino-7H-purin-7-yl)-4-fluoro-2,5-dihydrofuran-2-yl]oxy]methyl)phosphonic acid | - |
Human immunodeficiency virus 1 | |
([[(2S,5S)-5-(6-amino-7H-purin-7-yl)-2,5-dihydrofuran-2-yl]oxy]methyl)phosphonic acid | - |
Human immunodeficiency virus 1 | |
GS-9148 | 2'-Fd4AP | Human immunodeficiency virus 1 | |
Tenofovir | - |
Human immunodeficiency virus 1 |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Human immunodeficiency virus 1 | - |
- |
- |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
deoxynucleoside triphosphate + DNAn | - |
Human immunodeficiency virus 1 | diphosphate + DNAn+1 | - |
? |
Synonyms | Comment | Organism |
---|---|---|
reverse transcriptase | - |
Human immunodeficiency virus 1 |