Inhibitors | Comment | Organism | Structure |
---|---|---|---|
(+)-catechin | IC50: 0.44 mM | Gallus gallus | |
(-)-epicatechin | IC50: 0.32 mM | Gallus gallus | |
2,2'-Dihydroxychalcone | - |
Gallus gallus | |
3',4',5'-tri-O-methyltricetin | - |
Gallus gallus | |
3',4'-dihydroxyflavone | IC50: 0.262 mM | Gallus gallus | |
3,3',4'-trihydroxyflavone | IC50: 0.001 mM | Gallus gallus | |
5,4'-dihydroxyflavone | IC50: 0.024 mM | Gallus gallus | |
5,7-dihydroxyflavone | IC50: 0.043 mM | Gallus gallus | |
7,8,3',4'-tetrahydroxyflavone | IC50: 0.02 mM | Gallus gallus | |
7-O-methylapigenin | - |
Gallus gallus | |
apigenin | IC50: 0.023 mM | Gallus gallus | |
chalcone | - |
Gallus gallus | |
dihydroapigenin | IC50: 0.17 mM | Gallus gallus | |
dihydrofisetin | IC50: 0.18 mM | Gallus gallus | |
dihydroluteolin | - |
Gallus gallus | |
dihydroquercetin | IC50: 0.08 mM | Gallus gallus | |
fisetin | IC50: 0.005 mM | Gallus gallus | |
galangin | IC50: 0.02 mM | Gallus gallus | |
gossypol | - |
Gallus gallus | |
hesperidin | - |
Gallus gallus | |
isoliquiritigenin | - |
Gallus gallus | |
kaempferid | IC50: 0.008 mM | Gallus gallus | |
kaempferol | IC50: 0.004 mM | Gallus gallus | |
luteolin | IC50: 0.026 mM | Gallus gallus | |
additional information | no inhibition by epicatechin, pseudobabtisin, 4-dimethylaminobenzaldehyde | Gallus gallus | |
morin | IC50: 0.028 mM | Gallus gallus | |
myricetin | IC50: 0.006 mM | Gallus gallus | |
Okanin | - |
Gallus gallus | |
pseudobaptisin | - |
Gallus gallus | |
quercetagetin | IC50: 0.026 mM | Gallus gallus | |
quercetin | IC50: 0.006 mM | Gallus gallus | |
quercetrin | IC50: 0.137 mM | Gallus gallus | |
rutin | IC50: 0.32 mM | Gallus gallus | |
tricetin | IC50: 0.012 mM | Gallus gallus |
Metals/Ions | Comment | Organism | Structure |
---|---|---|---|
Ca2+ | - |
Gallus gallus |
Natural Substrates | Organism | Comment (Nat. Sub.) | Natural Products | Comment (Nat. Pro.) | Rev. | Reac. |
---|---|---|---|---|---|---|
ATP + myosin light chain | Gallus gallus | - |
ADP + myosin light chain phosphate | - |
? |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Gallus gallus | - |
- |
- |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
gizzard | - |
Gallus gallus | - |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
ATP + myosin light chain | - |
Gallus gallus | ADP + myosin light chain phosphate | - |
? |
Temperature Optimum [°C] | Temperature Optimum Maximum [°C] | Comment | Organism |
---|---|---|---|
30 | - |
assay at | Gallus gallus |
Cofactor | Comment | Organism | Structure |
---|---|---|---|
Calmodulin | requirement | Gallus gallus |
IC50 Value | IC50 Value Maximum | Comment | Organism | Inhibitor | Structure |
---|---|---|---|---|---|
0.001 | - |
IC50: 0.001 mM | Gallus gallus | 3,3',4'-trihydroxyflavone | |
0.004 | - |
IC50: 0.004 mM | Gallus gallus | kaempferol | |
0.005 | - |
IC50: 0.005 mM | Gallus gallus | fisetin | |
0.006 | - |
IC50: 0.006 mM | Gallus gallus | quercetin | |
0.006 | - |
IC50: 0.006 mM | Gallus gallus | myricetin | |
0.008 | - |
IC50: 0.008 mM | Gallus gallus | kaempferid | |
0.012 | - |
IC50: 0.012 mM | Gallus gallus | tricetin | |
0.02 | - |
IC50: 0.02 mM | Gallus gallus | galangin | |
0.02 | - |
IC50: 0.02 mM | Gallus gallus | 7,8,3',4'-tetrahydroxyflavone | |
0.023 | - |
IC50: 0.023 mM | Gallus gallus | apigenin | |
0.024 | - |
IC50: 0.024 mM | Gallus gallus | 5,4'-dihydroxyflavone | |
0.026 | - |
IC50: 0.026 mM | Gallus gallus | luteolin | |
0.026 | - |
IC50: 0.026 mM | Gallus gallus | quercetagetin | |
0.028 | - |
IC50: 0.028 mM | Gallus gallus | morin | |
0.043 | - |
IC50: 0.043 mM | Gallus gallus | 5,7-dihydroxyflavone | |
0.08 | - |
IC50: 0.08 mM | Gallus gallus | dihydroquercetin | |
0.137 | - |
IC50: 0.137 mM | Gallus gallus | quercetrin | |
0.17 | - |
IC50: 0.17 mM | Gallus gallus | dihydroapigenin | |
0.18 | - |
IC50: 0.18 mM | Gallus gallus | dihydrofisetin | |
0.262 | - |
IC50: 0.262 mM | Gallus gallus | 3',4'-dihydroxyflavone | |
0.32 | - |
IC50: 0.32 mM | Gallus gallus | rutin | |
0.32 | - |
IC50: 0.32 mM | Gallus gallus | (-)-epicatechin | |
0.44 | - |
IC50: 0.44 mM | Gallus gallus | (+)-catechin |