Inhibitors | Comment | Organism | Structure |
---|---|---|---|
(6R)-6-([[(1S)-1-(5-fluoro-2-methoxyphenyl)ethyl]amino]methyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide | - |
Homo sapiens | |
1-[(3R)-1-benzylpyrrolidin-3-yl]-3-[(3,5-dimethyl-1,2-oxazol-4-yl)methyl]urea | - |
Homo sapiens | |
2-[(2-amino-2-oxoethyl)(propan-2-yl)amino]-N-[(1S)-1-(naphthalen-2-yl)ethyl]acetamide | - |
Homo sapiens | |
2-[(3S)-3-[(phenylsulfanyl)methyl]pyrrolidin-1-yl]-N-(pyridin-3-ylmethyl)acetamide | - |
Homo sapiens | |
3-cyano-N-[[(3R)-1-(thiophen-2-ylmethyl)piperidin-3-yl]methyl]benzamide | - |
Homo sapiens | |
4-acetyl-N-[(2S)-2-(dimethylamino)-2-(4-methoxyphenyl)ethyl]-1H-pyrrole-2-carboxamide | - |
Homo sapiens | |
4-acetyl-N-[2-(3,4-dihydroisoquinolin-2(1H)-yl)-2-methylpropyl]-1H-pyrrole-2-carboxamide | - |
Homo sapiens | |
4-acetyl-N-[[(3R)-1-benzylpiperidin-3-yl]methyl]-1H-pyrrole-2-carboxamide | - |
Homo sapiens | |
5-(4-fluorophenyl)-N-[[(3S,5R,8aR)-hexahydro-1H-pyrrolo[2,1-c][1,4]oxazin-3-yl]methyl]-5-oxopentanamide | - |
Homo sapiens | |
5-fluoro-N-(imidazo[1,2-a]pyridin-2-ylmethyl)-2-methoxybenzamide | - |
Homo sapiens | |
CCG224406 | - |
Homo sapiens | |
CCG258208 | - |
Homo sapiens | |
GSK180736A | - |
Homo sapiens | |
N-(4-acetylphenyl)-N2-[(3-chlorophenyl)methyl]-N2-methyl-L-alaninamide | - |
Homo sapiens | |
N-(4-cyanophenyl)-3-[4-(4-hydroxyphenyl)-3,6-dihydropyridin-1(2H)-yl]propanamide | - |
Homo sapiens | |
N-[(2R)-2-(3,4-dihydroisoquinolin-2(1H)-yl)butyl]-N'-(1-ethyl-1H-pyrazol-4-yl)urea | - |
Homo sapiens | |
N-[(2R)-2-(3,4-dihydroisoquinolin-2(1H)-yl)propyl]-N'-[(2S)-1-(1H-pyrrol-1-yl)propan-2-yl]urea | - |
Homo sapiens | |
N-[1-[benzyl(methyl)amino]-2-methylpropan-2-yl]-6-methyl-4-oxo-1,4-dihydropyridine-3-carboxamide | - |
Homo sapiens | |
N2-methyl-N2-[[4-(methylsulfanyl)phenyl]methyl]-N-(1,3,5-trimethyl-1H-pyrazol-4-yl)-L-alaninamide | - |
Homo sapiens | |
N3-[(6-fluoroquinolin-8-yl)methyl]-N-[(pyridin-3-yl)methyl]-beta-alaninamide | - |
Homo sapiens | |
paroxetine | - |
Homo sapiens | |
Takeda CMPD 101 | - |
Homo sapiens | |
Takeda CMPD 103A | - |
Homo sapiens |
Natural Substrates | Organism | Comment (Nat. Sub.) | Natural Products | Comment (Nat. Pro.) | Rev. | Reac. |
---|---|---|---|---|---|---|
ATP + [beta-adrenergic receptor] | Homo sapiens | - |
ADP + phospho-[beta-adrenergic receptor] | - |
? |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | P25098 | - |
- |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
ATP + [beta-adrenergic receptor] | - |
Homo sapiens | ADP + phospho-[beta-adrenergic receptor] | - |
? |
Synonyms | Comment | Organism |
---|---|---|
G protein-coupled receptors kinase 2 | - |
Homo sapiens |
GRK2 | - |
Homo sapiens |