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Literature summary for 2.7.11.15 extracted from

  • Cannavo, A.; Liccardo, D.; Lymperopoulos, A.; Gambino, G.; DAmico, M.L.; Rengo, F.; Koch, W.J.; Leosco, D.; Ferrara, N.; Rengo, G.
    beta Adrenergic receptor kinase c-terminal peptide gene-therapy improves beta2-adrenergic receptor-dependent neoangiogenesis after hindlimb ischemia (2016), J. Pharmacol. Exp. Ther., 356, 503-513.
    View publication on PubMedView publication on EuropePMC

Inhibitors

Inhibitors Comment Organism Structure
beta adrenergic receptor kinase C-terminal peptide
-
Rattus norvegicus

Natural Substrates/ Products (Substrates)

Natural Substrates Organism Comment (Nat. Sub.) Natural Products Comment (Nat. Pro.) Rev. Reac.
ATP + [beta-adrenergic receptor] Rattus norvegicus
-
ADP + phospho-[beta-adrenergic receptor]
-
?

Organism

Organism UniProt Comment Textmining
Rattus norvegicus
-
-
-

Source Tissue

Source Tissue Comment Organism Textmining
skeletal muscle
-
Rattus norvegicus
-

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
ATP + [beta-adrenergic receptor]
-
Rattus norvegicus ADP + phospho-[beta-adrenergic receptor]
-
?

Synonyms

Synonyms Comment Organism
G protein-coupled receptor kinase 2
-
Rattus norvegicus
GRK2
-
Rattus norvegicus

Expression

Organism Comment Expression
Rattus norvegicus 15 days of ischemia result in 2-fold increase in enzyme levels in the ischemic muscle down