Protein Variants | Comment | Organism |
---|---|---|
C199A | inactive | Mus musculus |
Inhibitors | Comment | Organism | Structure |
---|---|---|---|
myr-PKI(14-22) | reversible inhibitor | Mus musculus | |
rhodamine B-PKI(14-22)-GFMK | potent, competitive, irreversible inhibitor, 97% inhibition at 0.001 mM | Mus musculus |
Natural Substrates | Organism | Comment (Nat. Sub.) | Natural Products | Comment (Nat. Pro.) | Rev. | Reac. |
---|---|---|---|---|---|---|
ATP + a protein | Mus musculus | - |
ADP + phosphorylated protein | - |
? |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Mus musculus | P05132 | - |
- |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
ATP + a protein | - |
Mus musculus | ADP + phosphorylated protein | - |
? |
Synonyms | Comment | Organism |
---|---|---|
cAMP-dependent protein kinase | - |
Mus musculus |
PKACalpha | catalytic subunit | Mus musculus |
IC50 Value | IC50 Value Maximum | Comment | Organism | Inhibitor | Structure |
---|---|---|---|---|---|
0.0000118 | - |
pH and temperature not specified in the publication | Mus musculus | rhodamine B-PKI(14-22)-GFMK | |
0.0000479 | - |
pH and temperature not specified in the publication | Mus musculus | myr-PKI(14-22) |