Inhibitors | Comment | Organism | Structure |
---|---|---|---|
B-5354c | SPHK1, SPHK2, noncompetitive to sphingosine | Homo sapiens | |
F-12509A | SPHK1, SPHK2, competitive to sphingosine | Homo sapiens | |
N,N-dimethylsphingosine | - |
Homo sapiens |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | - |
recombinant SPHK1, SPHK2 | - |
Ki Value [mM] | Ki Value maximum [mM] | Inhibitor | Comment | Organism | Structure |
---|---|---|---|---|---|
0.0022 | - |
B-5354c | SPHK2 | Homo sapiens | |
0.003 | - |
N,N-dimethylsphingosine | SPHK1 | Homo sapiens | |
0.004 | - |
F-12509A | SPHK1 | Homo sapiens | |
0.004 | - |
B-5354c | SPHK1 | Homo sapiens | |
0.0055 | - |
F-12509A | SPHK2 | Homo sapiens | |
0.0086 | - |
N,N-dimethylsphingosine | SPHK2 | Homo sapiens |