Crystallization (Comment) | Organism |
---|---|
cytosolic isoform in complex with gabapentin or 4-methylvalerate, mitochondrial isoform in complex with gabapentin | Homo sapiens |
Inhibitors | Comment | Organism | Structure |
---|---|---|---|
gabapentin | inhibition is isoform-specific | Homo sapiens |
Localization | Comment | Organism | GeneOntology No. | Textmining |
---|---|---|---|---|
cytosol | - |
Homo sapiens | 5829 | - |
mitochondrion | - |
Homo sapiens | 5739 | - |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | O15382 | cytosolic and mitochondrial isoforms | - |
Cofactor | Comment | Organism | Structure |
---|---|---|---|
pyridoxal 5'-phosphate | - |
Homo sapiens |
Ki Value [mM] | Ki Value maximum [mM] | Inhibitor | Comment | Organism | Structure |
---|---|---|---|---|---|
1.3 | - |
gabapentin | cytosolic isoform, reduced | Homo sapiens | |
3.5 | - |
gabapentin | cytosolic isoform, oxidized | Homo sapiens | |
65.4 | - |
gabapentin | mitochondrial isoform, reduced | Homo sapiens | |
389.2 | - |
gabapentin | mitochondrial isoform, oxidized | Homo sapiens |