Cloned (Comment) | Organism |
---|---|
expressed in Escherichia coli BL21(DE3) cells | Paenibacillus larvae subsp. larvae |
Crystallization (Comment) | Organism |
---|---|
hanging drop vapor diffusion method, using 28% (w/v) PEG 4000, 200 mM sodium acetate, and 100 mM Tris, pH 8.5 | Paenibacillus larvae subsp. larvae |
Inhibitors | Comment | Organism | Structure |
---|---|---|---|
N-[[1-(1H-pyrazolo[3,4-d]pyrimidin-4-yl)piperidin-3-yl]methyl]methanesulfonamide | - |
Paenibacillus larvae subsp. larvae |
KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.017 | - |
(ADP-D-ribosyl)n-RhoA protein | at pH 7.4 and 37°C | Paenibacillus larvae subsp. larvae | |
0.034 | - |
NAD+ | at pH 7.4 and 37°C | Paenibacillus larvae subsp. larvae |
Molecular Weight [Da] | Molecular Weight Maximum [Da] | Comment | Organism |
---|---|---|---|
22000 | - |
x * 22000, calculated from amino acid sequence | Paenibacillus larvae subsp. larvae |
Natural Substrates | Organism | Comment (Nat. Sub.) | Natural Products | Comment (Nat. Pro.) | Rev. | Reac. |
---|---|---|---|---|---|---|
NAD+ + (ADP-D-ribosyl)n-RhoA protein | Paenibacillus larvae subsp. larvae | - |
nicotinamide + (ADP-D-ribosyl)n+1-RhoA protein + H+ | - |
? | |
NAD+ + (ADP-D-ribosyl)n-RhoA protein | Paenibacillus larvae subsp. larvae BRL-230010 | - |
nicotinamide + (ADP-D-ribosyl)n+1-RhoA protein + H+ | - |
? |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Paenibacillus larvae subsp. larvae | W2E3J5 | - |
- |
Paenibacillus larvae subsp. larvae BRL-230010 | W2E3J5 | - |
- |
Purification (Comment) | Organism |
---|---|
HiTrap chelating Sepharose column chromatography, and Superdex 200 gel filtration | Paenibacillus larvae subsp. larvae |
Source Tissue | Comment | Organism | Textmining |
---|
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
NAD+ + (ADP-D-ribosyl)n-RhoA protein | - |
Paenibacillus larvae subsp. larvae | nicotinamide + (ADP-D-ribosyl)n+1-RhoA protein + H+ | - |
? | |
NAD+ + (ADP-D-ribosyl)n-RhoA protein | - |
Paenibacillus larvae subsp. larvae BRL-230010 | nicotinamide + (ADP-D-ribosyl)n+1-RhoA protein + H+ | - |
? |
Subunits | Comment | Organism |
---|---|---|
? | x * 22000, calculated from amino acid sequence | Paenibacillus larvae subsp. larvae |
Synonyms | Comment | Organism |
---|---|---|
ADP-ribosyltransferase | - |
Paenibacillus larvae subsp. larvae |
C3larvin toxin | - |
Paenibacillus larvae subsp. larvae |
Ki Value [mM] | Ki Value maximum [mM] | Inhibitor | Comment | Organism | Structure |
---|---|---|---|---|---|
0.011 | - |
N-[[1-(1H-pyrazolo[3,4-d]pyrimidin-4-yl)piperidin-3-yl]methyl]methanesulfonamide | at pH 7.4 and 37°C | Paenibacillus larvae subsp. larvae |
Organism | Comment | pI Value Maximum | pI Value |
---|---|---|---|
Paenibacillus larvae subsp. larvae | calculated from amino acid sequence | - |
9.6 |