Inhibitors | Comment | Organism | Structure |
---|---|---|---|
8-aza-2,6-diaminopurine | noncompetitive | Oryctolagus cuniculus | |
aminopterin | noncompetitive | Oryctolagus cuniculus | |
D,L-6-methyl 5,6,7,8-tetrahydropterin | competitive | Oryctolagus cuniculus | |
erythro-9-(2-hydroxy-3-nonyl)adenine | competitive | Oryctolagus cuniculus | |
folate | competitive | Oryctolagus cuniculus | |
PCMB | 0.1 mM, 85% loss of activity within 15 min | Oryctolagus cuniculus |
KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.06 | - |
guanosine | - |
Oryctolagus cuniculus |
Molecular Weight [Da] | Molecular Weight Maximum [Da] | Comment | Organism |
---|---|---|---|
70000 | - |
gel filtration | Oryctolagus cuniculus |
345000 | - |
2 * 345000, SDS-PAGE | Oryctolagus cuniculus |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Oryctolagus cuniculus | - |
- |
- |
Oxidation Stability | Organism |
---|---|
high sensitivity to photooxidation in presence of methylene blue, almost 95% loss of activity after 40 min irradiation | Oryctolagus cuniculus |
Purification (Comment) | Organism |
---|---|
- |
Oryctolagus cuniculus |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
brain | - |
Oryctolagus cuniculus | - |
Specific Activity Minimum [µmol/min/mg] | Specific Activity Maximum [µmol/min/mg] | Comment | Organism |
---|---|---|---|
50 | - |
- |
Oryctolagus cuniculus |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
guanosine + phosphate | - |
Oryctolagus cuniculus | guanine + alpha-D-ribose 1-phosphate | - |
? |
Subunits | Comment | Organism |
---|---|---|
dimer | 2 * 345000, SDS-PAGE | Oryctolagus cuniculus |
Ki Value [mM] | Ki Value maximum [mM] | Inhibitor | Comment | Organism | Structure |
---|---|---|---|---|---|
0.0337 | - |
folic acid | - |
Oryctolagus cuniculus | |
0.038 | - |
2-amino-6-methyl-5,6,7,8-tetrahydropteridin-4(1H)-one | - |
Oryctolagus cuniculus | |
0.15 | - |
aminopterin | - |
Oryctolagus cuniculus | |
0.19 | - |
erythro-9-(2-hydroxy-3-nonyl)adenine | - |
Oryctolagus cuniculus | |
0.195 | - |
8-aza-2,6-diaminopurine | - |
Oryctolagus cuniculus |