Literature summary for 2.3.1.82 extracted from

Gao, F.; Yan, X.; Baettig, O.M.; Berghuis, A.M.; Auclair, K.
Regio- and chemoselective 6-N-derivatization of amino-glycosides: bi-substrate inhibitors as probes to study amino-glycoside 6-N-acetyltransferase (2005), Angew. Chem. Int. Ed. Engl., 44, 6859-6862.

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Inhibitors

Inhibitors	Comment	Organism	Structure
CoA-aminoglycoside 1	-	Enterococcus faecium
CoA-aminoglycoside 11a	-	Enterococcus faecium
CoA-aminoglycoside 11b	-	Enterococcus faecium
CoA-aminoglycoside 11c	-	Enterococcus faecium
CoA-aminoglycoside 2	-	Enterococcus faecium
CoA-aminoglycoside 3	-	Enterococcus faecium

Organism

Organism	UniProt	Comment	Textmining
Enterococcus faecium	-	-	-

Ki Value [mM]

Ki Value [mM]	Ki Value maximum [mM]	Inhibitor	Comment	Organism	Structure
0.000043	-	CoA-aminoglycoside 11a	-	Enterococcus faecium
0.000076	-	CoA-aminoglycoside 1	-	Enterococcus faecium
0.000111	-	CoA-aminoglycoside 2	-	Enterococcus faecium
0.000119	-	CoA-aminoglycoside 3	-	Enterococcus faecium
0.000161	-	CoA-aminoglycoside 11b	-	Enterococcus faecium
0.00799	-	CoA-aminoglycoside 11c	-	Enterococcus faecium

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Release 2023.1 (January 2023)