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Literature summary for 1.5.1.3 extracted from

  • Ferone, R.
    Dihydrofolate reductase from pyrimethamine-resistant Plasmodium berghei (1970), J. Biol. Chem., 245, 850-854.
    View publication on PubMed

Inhibitors

Inhibitors Comment Organism Structure
pyrimethamine
-
Plasmodium berghei
trimethoprim
-
Plasmodium berghei

KM Value [mM]

KM Value [mM] KM Value Maximum [mM] Substrate Comment Organism Structure
additional information
-
additional information
-
Plasmodium berghei

Metals/Ions

Metals/Ions Comment Organism Structure
K+ stimulation Plasmodium berghei

Organism

Organism UniProt Comment Textmining
Plasmodium berghei
-
pyrimethamine-sensitive and pyrimethamine-resistant strain
-

Turnover Number [1/s]

Turnover Number Minimum [1/s] Turnover Number Maximum [1/s] Substrate Comment Organism Structure
additional information
-
additional information pyrimethamine sensitive and resistant strain Plasmodium berghei

Ki Value [mM]

Ki Value [mM] Ki Value maximum [mM] Inhibitor Comment Organism Structure
0.00000037
-
pyrimethamine trimethoprim-sensitive strain Plasmodium berghei
0.0000071
-
trimethoprim trimethoprim-sensitive strain Plasmodium berghei
0.000014
-
pyrimethamine trimethoprim-resistant sdtrain Plasmodium berghei
0.000068
-
trimethoprim trimethoprim-resistant strain Plasmodium berghei