Cloned (Comment) | Organism |
---|---|
expression in Escherichia coli | Cereibacter sphaeroides |
Protein Variants | Comment | Organism |
---|---|---|
G95S | marginal increase in resistance to diazaborine | Cereibacter sphaeroides |
P155Q | strong increase in resistance to diazaborine | Cereibacter sphaeroides |
Inhibitors | Comment | Organism | Structure |
---|---|---|---|
diazaborine | 0.019 mM, 50% inhibition of wild-type FabI1, 0.25 mM, 50% inhibition of P155Q mutant FabI1 | Cereibacter sphaeroides | |
triclosan | 0.01 mM, 50% inhibition of wild-type FabI1, 0.15 mM, 50% inhibition of P155Q mutant FabI1 | Cereibacter sphaeroides |
KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.021 | - |
NADH | 30°C, pH 6.5 | Cereibacter sphaeroides | |
1.6 | - |
trans-but-2-enoyl-[acyl-carrier protein] | 30°C, pH 6.5 | Cereibacter sphaeroides |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Cereibacter sphaeroides | - |
- |
- |
Purification (Comment) | Organism |
---|---|
recombinant FabI1 | Cereibacter sphaeroides |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
trans-but-2-enoyl-[acyl-carrier protein] + NADH | - |
Cereibacter sphaeroides | butanoyl-[acyl-carrier protein] + NAD+ | - |
? |
Synonyms | Comment | Organism |
---|---|---|
enoyl-acyl carrier protein reductase | - |
Cereibacter sphaeroides |
FabI1 | - |
Cereibacter sphaeroides |
Turnover Number Minimum [1/s] | Turnover Number Maximum [1/s] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.48 | - |
trans-but-2-enoyl-[acyl-carrier protein] | 30°C, pH 6.5, G95S mutant | Cereibacter sphaeroides | |
0.65 | - |
trans-but-2-enoyl-[acyl-carrier protein] | 30°C, pH 6.5 | Cereibacter sphaeroides | |
1 | - |
trans-but-2-enoyl-[acyl-carrier protein] | 30°C, pH 6.5, P155Q mutant | Cereibacter sphaeroides |
Cofactor | Comment | Organism | Structure |
---|---|---|---|
NADH | - |
Cereibacter sphaeroides |
Ki Value [mM] | Ki Value maximum [mM] | Inhibitor | Comment | Organism | Structure |
---|---|---|---|---|---|
0.002 | - |
triclosane | 30°C, pH 6.5 | Cereibacter sphaeroides | |
0.008 | - |
triclosane | 30°C, pH 6.5, G95S mutant | Cereibacter sphaeroides | |
0.0084 | - |
diazaborine | 30°C, pH 6.5 | Cereibacter sphaeroides | |
0.03 | - |
diazaborine | 30°C, pH 6.5, G95S mutant | Cereibacter sphaeroides | |
0.18 | - |
triclosane | 30°C, pH 6.5, P155Q mutant | Cereibacter sphaeroides | |
0.29 | - |
diazaborine | 30°C, pH 6.5, P155Q mutant | Cereibacter sphaeroides |