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Literature summary for 1.3.1.9 extracted from

  • Muench, S.P.; Rafferty, J.B.; McLeod, R.; Rice, D.W.; Prigge, S.T.
    Expression, purification and crystallization of the Plasmodium falciparum enoyl reductase (2003), Acta Crystallogr. Sect. D, 59, 1246-1248.
    View publication on PubMed

Cloned(Commentary)

Cloned (Comment) Organism
expression in Escherichia coli Plasmodium falciparum

Crystallization (Commentary)

Crystallization (Comment) Organism
crystals are grown by hanging-drop vapour-diffusion, 0.0025 ml protein solution containing 12 mg/ml enzyme in 20 mM sodium/potassium phosphate, pH 8.0, 150 mM NaCl, 0.005 mM NAD+ and 0.006 mM triclosan are mixed with 0.0025 ml reservoir solution at 17°C, optimal reservoir solution contains 19.5% polyethylene glycol 3350 and 230 mM KI, crystals diffract to 2.2 A Plasmodium falciparum

Inhibitors

Inhibitors Comment Organism Structure
triclosan
-
Plasmodium falciparum

Organism

Organism UniProt Comment Textmining
Plasmodium falciparum
-
-
-

Purification (Commentary)

Purification (Comment) Organism
recombinant His-tagged pfENR Plasmodium falciparum

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
acyl-[acyl-carrier protein] + NAD+
-
Plasmodium falciparum trans-2,3-dehydroacyl-[acyl-carrier protein] + NADH
-
?

Synonyms

Synonyms Comment Organism
pfENR
-
Plasmodium falciparum

Cofactor

Cofactor Comment Organism Structure
NAD+
-
Plasmodium falciparum