Cloned (Comment) | Organism |
---|---|
expression in Escherichia coli | Mycolicibacterium smegmatis |
Protein Variants | Comment | Organism |
---|---|---|
additional information | isolation of mutant strains resistant to dinitrobenzamides. All mutants show cross-resistance to benzothiazinones and dinitrobenzamides, and all the mutant strains with a higher level of resistance to dinitrobenzamides have a substitution C394G of MSMEG_6382 gene encoding decaprenylphospho-?-D-ribofuranose 2-oxidase | Mycolicibacterium smegmatis |
Inhibitors | Comment | Organism | Structure |
---|---|---|---|
additional information | benzothiazinone and dinitrobenzamide inhibitors target decaprenylphospho-beta-D-ribofuranose 2-oxidase DprE1. Several mutants showing high levels of dinitrobenzamide resistance, exhibit a mutation in residue Cys394 of DprE1 | Mycolicibacterium smegmatis |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Mycolicibacterium smegmatis | A0R607 | - |
- |
Synonyms | Comment | Organism |
---|---|---|
DprE2 | - |
Mycolicibacterium smegmatis |
MSMEG_6382 | - |
Mycolicibacterium smegmatis |