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Literature summary for 1.1.1.184 extracted from

  • Imamura, Y.; Shimada, H.
    Differential pharmacokinetics of acetohexamide in male Wistar-Imamichi and Sprague-Dawley rats: role of microsomal carbonyl reductase (2005), Biol. Pharm. Bull., 28, 185-187.
    View publication on PubMed

KM Value [mM]

KM Value [mM] KM Value Maximum [mM] Substrate Comment Organism Structure
additional information
-
additional information pharmacokinetics of acetohexamide in male Wistar-Imamichi, showing very low enzyme amount, and Sprague-Dawley rats, overview Rattus norvegicus

Localization

Localization Comment Organism GeneOntology No. Textmining
microsome
-
Rattus norvegicus
-
-

Organism

Organism UniProt Comment Textmining
Rattus norvegicus
-
male Wistar-Imamichi, showing very low enzyme amount, and Sprague-Dawley rats
-

Specific Activity [micromol/min/mg]

Specific Activity Minimum [µmol/min/mg] Specific Activity Maximum [µmol/min/mg] Comment Organism
additional information
-
plasma clearance of acetohexamide in male Wistar-Imamichi, showing very low enzyme amount, and Sprague-Dawley rats, overview Rattus norvegicus

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
acetohexamide + NADPH + H+
-
Rattus norvegicus ?
-
?

Synonyms

Synonyms Comment Organism
microsomal carbonyl reductase
-
Rattus norvegicus

pH Optimum

pH Optimum Minimum pH Optimum Maximum Comment Organism
6.5
-
assay at Rattus norvegicus

Cofactor

Cofactor Comment Organism Structure
NADPH
-
Rattus norvegicus