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0.0123 - 0.03
(4Z,7E)-N,N'-dihydroxy-2,2-dimethyl-5,6-dihydro-2H-benzimidazole-4,7-diimine
0.0033 - 0.0418
(5Z)-2-amino-5-(2-nitrobenzylidene)-1,3-thiazol-4(5H)-one
0.0038 - 0.012
1,4-dioxo-1,2,3,4-tetrahydronaphthalen-2-yl 2,3,4-tri-O-acetylpentopyranoside
0.0055 - 0.0142
1-(2-nitrobenzyl)-1H-indole-3-carbaldehyde
0.002 - 4
10H-indeno[2,1-e]tetrazolo[1,5-b][1,2,4]triazin-10-one
0.0051 - 0.1
2,4-bis[2-(4-hydroxyphenyl)propan-2-yl]phenol
0.0073 - 0.0209
2-(benzylsulfanyl)-3-(morpholin-4-yl)-2,3-dihydronaphthalene-1,4-dione
0.0052 - 0.1
2-chloro-N-[5-([2-oxo-2-[(4-sulfamoylphenyl)amino]ethyl]sulfanyl)-1,3,4-thiadiazol-2-yl]acetamide
0.0042 - 0.0108
2-hydroxy-2-(2-hydroxy-6-oxocyclohex-2-en-1-yl)-1H-indene-1,3(2H)-dione
0.0075 - 0.014
2-thioxo-3-[(E)-(3,3,5-trimethylcyclohexylidene)amino]-1,3-thiazolidin-4-one
0.0165 - 0.1
2-[(2-chloro-5-nitrobenzoyl)amino]-5-iodobenzoic acid
0.0082 - 0.014
2-[(3-formyl-1H-indol-1-yl)methyl]benzonitrile
0.0002 - 0.0212
3,3'-(4H-1,2,4-triazole-3,5-diyl)bis(4-nitro-1,2,5-oxadiazole)
0.0123
3-Mercaptopropionic acid
0.0202 - 0.1
3-[(2E)-2-[1-(3,4-dimethoxyphenyl)ethylidene]hydrazinyl]benzoic acid
0.0063 - 0.0122
3-[(E)-(2,6-difluorobenzylidene)amino]-2-thioxo-1,3-thiazolidin-4-one
0.0072 - 0.099
4,4'-(phenylmethanediyl)bis[2-(4-chlorophenyl)-5-methyl-2,4-dihydro-3H-pyrazol-3-one]
0.013 - 0.0226
4,4'-[(4-hydroxyphenyl)methanediyl]bis(2-heptyl-5-methyl-2,4-dihydro-3H-pyrazol-3-one)
0.0029 - 0.0045
4-(morpholin-4-yl)naphthalene-1,2-dione
0.003 - 0.0053
4-(piperidin-1-yl)naphthalene-1,2-dione
0.0034 - 0.065
4-nitro-1,6-dihydrobenzo[1,2-d:3,4-d']bis[1,2,3]triazole
0.0055 - 0.1
4-nitro-7-[[(1-phenyl-1H-tetrazol-5-yl)sulfanyl]methyl]-2,1,3-benzothiadiazole
0.0026 - 0.0112
4-[(1,4-dioxo-1,2,3,4-tetrahydronaphthalen-2-yl)sulfanyl]butanoic acid
0.0033 - 0.0083
5,6-dichloro-2,1,3-benzothiadiazole-4,7-diol
0.0069 - 0.0104
5-[(E)-benzylideneamino]-6-[(2-hydroxyethyl)amino]pyrimidine-2,4(1H,3H)-dione
0.0059 - 0.0129
5-[(E)-[[1-(2-chlorobenzyl)-1H-indol-3-yl]methylidene]amino]-1,3-dihydro-2H-benzimidazol-2-one
0.0122 - 0.0593
5-[[5-hydroxy-3-methyl-1-(4-methylphenyl)-1H-pyrazol-4-yl]methylidene]-1,3-diphenyl-2-thioxodihydropyrimidine-4,6(1H,5H)-dione
0.0021 - 0.0057
6,11-dioxo-5a,6,11,11a-tetrahydronaphtho[2',3':4,5][1,3]thiazolo[3,2-a]pyridin-12-ium
0.0045 - 0.1
9H-indeno[1,2-b][1,2,5]oxadiazolo[3,4-e]pyrazin-9-one
0.0049 - 0.0063
biphenyl-3,3'-dicarbaldehyde
0.0004 - 0.001
carboxymethoxylamine
0.001 - 4
methyl 2-amino-3-oxo-3H-phenothiazine-1-carboxylate
0.005 - 0.0125
methyl 2-[[(2-methylimidazo[1,2-a]pyridin-3-yl)carbonyl]amino]benzoate
0.0076 - 0.0164
N-(2-hydroxy-1,3-dioxo-2,3-dihydro-1H-inden-2-yl)benzamide
0.001 - 0.0022
N-[4,7-dioxo-6-(phenylamino)-4,7-dihydro-2,1,3-benzoxadiazol-5-yl]acetamide
0.0013 - 0.0044
N-[4,7-dioxo-6-(piperidin-1-yl)-4,7-dihydro-2,1,3-benzoxadiazol-5-yl]acetamide
0.0037 - 0.0591
naphtho[2',3':4,5]imidazo[1,2-a]pyridine-6,11-dione
0.0244 - 0.1
[(1,3-dioxo-1,3-dihydro-2H-isoindol-2-yl)oxy]acetic acid
0.0123
(4Z,7E)-N,N'-dihydroxy-2,2-dimethyl-5,6-dihydro-2H-benzimidazole-4,7-diimine
Mus musculus
pH 8.0, 37°C, recombinant enzyme
0.0135
(4Z,7E)-N,N'-dihydroxy-2,2-dimethyl-5,6-dihydro-2H-benzimidazole-4,7-diimine
Rhipicephalus microplus
pH 8.0, 37°C, recombinant enzyme
0.0266
(4Z,7E)-N,N'-dihydroxy-2,2-dimethyl-5,6-dihydro-2H-benzimidazole-4,7-diimine
Mus musculus
pH 8.0, 37°C, recombinant enzyme
0.0274
(4Z,7E)-N,N'-dihydroxy-2,2-dimethyl-5,6-dihydro-2H-benzimidazole-4,7-diimine
Ctenocephalides felis
pH 8.0, 37°C, recombinant enzyme
0.03
(4Z,7E)-N,N'-dihydroxy-2,2-dimethyl-5,6-dihydro-2H-benzimidazole-4,7-diimine
Drosophila melanogaster
pH 8.0, 37°C, recombinant enzyme
0.0033
(5Z)-2-amino-5-(2-nitrobenzylidene)-1,3-thiazol-4(5H)-one
Drosophila melanogaster
pH 8.0, 37°C, recombinant enzyme
0.0033
(5Z)-2-amino-5-(2-nitrobenzylidene)-1,3-thiazol-4(5H)-one
Mus musculus
pH 8.0, 37°C, recombinant enzyme
0.0037
(5Z)-2-amino-5-(2-nitrobenzylidene)-1,3-thiazol-4(5H)-one
Ctenocephalides felis
pH 8.0, 37°C, recombinant enzyme
0.0057
(5Z)-2-amino-5-(2-nitrobenzylidene)-1,3-thiazol-4(5H)-one
Rhipicephalus microplus
pH 8.0, 37°C, recombinant enzyme
0.0418
(5Z)-2-amino-5-(2-nitrobenzylidene)-1,3-thiazol-4(5H)-one
Mus musculus
pH 8.0, 37°C, recombinant enzyme
0.0038
1,4-dioxo-1,2,3,4-tetrahydronaphthalen-2-yl 2,3,4-tri-O-acetylpentopyranoside
Drosophila melanogaster
pH 8.0, 37°C, recombinant enzyme
0.004
1,4-dioxo-1,2,3,4-tetrahydronaphthalen-2-yl 2,3,4-tri-O-acetylpentopyranoside
Rhipicephalus microplus
pH 8.0, 37°C, recombinant enzyme
0.004
1,4-dioxo-1,2,3,4-tetrahydronaphthalen-2-yl 2,3,4-tri-O-acetylpentopyranoside
Mus musculus
pH 8.0, 37°C, recombinant enzyme
0.0053
1,4-dioxo-1,2,3,4-tetrahydronaphthalen-2-yl 2,3,4-tri-O-acetylpentopyranoside
Ctenocephalides felis
pH 8.0, 37°C, recombinant enzyme
0.012
1,4-dioxo-1,2,3,4-tetrahydronaphthalen-2-yl 2,3,4-tri-O-acetylpentopyranoside
Mus musculus
pH 8.0, 37°C, recombinant enzyme
0.0055
1-(2-nitrobenzyl)-1H-indole-3-carbaldehyde
Ctenocephalides felis
pH 8.0, 37°C, recombinant enzyme
0.0069
1-(2-nitrobenzyl)-1H-indole-3-carbaldehyde
Mus musculus
pH 8.0, 37°C, recombinant enzyme
0.0076
1-(2-nitrobenzyl)-1H-indole-3-carbaldehyde
Drosophila melanogaster
pH 8.0, 37°C, recombinant enzyme
0.008
1-(2-nitrobenzyl)-1H-indole-3-carbaldehyde
Rhipicephalus microplus
pH 8.0, 37°C, recombinant enzyme
0.0142
1-(2-nitrobenzyl)-1H-indole-3-carbaldehyde
Mus musculus
pH 8.0, 37°C, recombinant enzyme
0.002
10H-indeno[2,1-e]tetrazolo[1,5-b][1,2,4]triazin-10-one
Rhipicephalus microplus
pH 8.0, 37°C, recombinant enzyme
0.002
10H-indeno[2,1-e]tetrazolo[1,5-b][1,2,4]triazin-10-one
Drosophila melanogaster
pH 8.0, 37°C, recombinant enzyme
0.002
10H-indeno[2,1-e]tetrazolo[1,5-b][1,2,4]triazin-10-one
Mus musculus
pH 8.0, 37°C, recombinant enzyme
0.002 - 4
10H-indeno[2,1-e]tetrazolo[1,5-b][1,2,4]triazin-10-one
Ctenocephalides felis
pH 8.0, 37°C, recombinant enzyme
0.0047
10H-indeno[2,1-e]tetrazolo[1,5-b][1,2,4]triazin-10-one
Mus musculus
pH 8.0, 37°C, recombinant enzyme
0.0051
2,4-bis[2-(4-hydroxyphenyl)propan-2-yl]phenol
Rhipicephalus microplus
pH 8.0, 37°C, recombinant enzyme
0.0777
2,4-bis[2-(4-hydroxyphenyl)propan-2-yl]phenol
Mus musculus
pH 8.0, 37°C, recombinant enzyme
0.1
2,4-bis[2-(4-hydroxyphenyl)propan-2-yl]phenol
Mus musculus
above, pH 8.0, 37°C, recombinant enzyme
0.1
2,4-bis[2-(4-hydroxyphenyl)propan-2-yl]phenol
Ctenocephalides felis
above, pH 8.0, 37°C, recombinant enzyme
0.1
2,4-bis[2-(4-hydroxyphenyl)propan-2-yl]phenol
Drosophila melanogaster
above, pH 8.0, 37°C, recombinant enzyme
0.0073
2-(benzylsulfanyl)-3-(morpholin-4-yl)-2,3-dihydronaphthalene-1,4-dione
Mus musculus
pH 8.0, 37°C, recombinant enzyme
0.0089
2-(benzylsulfanyl)-3-(morpholin-4-yl)-2,3-dihydronaphthalene-1,4-dione
Drosophila melanogaster
pH 8.0, 37°C, recombinant enzyme
0.0112
2-(benzylsulfanyl)-3-(morpholin-4-yl)-2,3-dihydronaphthalene-1,4-dione
Rhipicephalus microplus
pH 8.0, 37°C, recombinant enzyme
0.0115
2-(benzylsulfanyl)-3-(morpholin-4-yl)-2,3-dihydronaphthalene-1,4-dione
Ctenocephalides felis
pH 8.0, 37°C, recombinant enzyme
0.0209
2-(benzylsulfanyl)-3-(morpholin-4-yl)-2,3-dihydronaphthalene-1,4-dione
Mus musculus
pH 8.0, 37°C, recombinant enzyme
0.0052
2-chloro-N-[5-([2-oxo-2-[(4-sulfamoylphenyl)amino]ethyl]sulfanyl)-1,3,4-thiadiazol-2-yl]acetamide
Mus musculus
pH 8.0, 37°C, recombinant enzyme
0.0087
2-chloro-N-[5-([2-oxo-2-[(4-sulfamoylphenyl)amino]ethyl]sulfanyl)-1,3,4-thiadiazol-2-yl]acetamide
Mus musculus
pH 8.0, 37°C, recombinant enzyme
0.0162
2-chloro-N-[5-([2-oxo-2-[(4-sulfamoylphenyl)amino]ethyl]sulfanyl)-1,3,4-thiadiazol-2-yl]acetamide
Ctenocephalides felis
pH 8.0, 37°C, recombinant enzyme
0.0284
2-chloro-N-[5-([2-oxo-2-[(4-sulfamoylphenyl)amino]ethyl]sulfanyl)-1,3,4-thiadiazol-2-yl]acetamide
Drosophila melanogaster
pH 8.0, 37°C, recombinant enzyme
0.1
2-chloro-N-[5-([2-oxo-2-[(4-sulfamoylphenyl)amino]ethyl]sulfanyl)-1,3,4-thiadiazol-2-yl]acetamide
Rhipicephalus microplus
above, pH 8.0, 37°C, recombinant enzyme
0.0042
2-hydroxy-2-(2-hydroxy-6-oxocyclohex-2-en-1-yl)-1H-indene-1,3(2H)-dione
Mus musculus
pH 8.0, 37°C, recombinant enzyme
0.0047
2-hydroxy-2-(2-hydroxy-6-oxocyclohex-2-en-1-yl)-1H-indene-1,3(2H)-dione
Drosophila melanogaster
pH 8.0, 37°C, recombinant enzyme
0.0062
2-hydroxy-2-(2-hydroxy-6-oxocyclohex-2-en-1-yl)-1H-indene-1,3(2H)-dione
Ctenocephalides felis
pH 8.0, 37°C, recombinant enzyme
0.0069
2-hydroxy-2-(2-hydroxy-6-oxocyclohex-2-en-1-yl)-1H-indene-1,3(2H)-dione
Rhipicephalus microplus
pH 8.0, 37°C, recombinant enzyme
0.0108
2-hydroxy-2-(2-hydroxy-6-oxocyclohex-2-en-1-yl)-1H-indene-1,3(2H)-dione
Mus musculus
pH 8.0, 37°C, recombinant enzyme
0.0075
2-thioxo-3-[(E)-(3,3,5-trimethylcyclohexylidene)amino]-1,3-thiazolidin-4-one
Rhipicephalus microplus
pH 8.0, 37°C, recombinant enzyme
0.01
2-thioxo-3-[(E)-(3,3,5-trimethylcyclohexylidene)amino]-1,3-thiazolidin-4-one
Mus musculus
pH 8.0, 37°C, recombinant enzyme
0.0127
2-thioxo-3-[(E)-(3,3,5-trimethylcyclohexylidene)amino]-1,3-thiazolidin-4-one
Mus musculus
pH 8.0, 37°C, recombinant enzyme
0.0139
2-thioxo-3-[(E)-(3,3,5-trimethylcyclohexylidene)amino]-1,3-thiazolidin-4-one
Ctenocephalides felis
pH 8.0, 37°C, recombinant enzyme
0.014
2-thioxo-3-[(E)-(3,3,5-trimethylcyclohexylidene)amino]-1,3-thiazolidin-4-one
Drosophila melanogaster
pH 8.0, 37°C, recombinant enzyme
0.0165
2-[(2-chloro-5-nitrobenzoyl)amino]-5-iodobenzoic acid
Ctenocephalides felis
pH 8.0, 37°C, recombinant enzyme
0.0714
2-[(2-chloro-5-nitrobenzoyl)amino]-5-iodobenzoic acid
Drosophila melanogaster
pH 8.0, 37°C, recombinant enzyme
0.0845
2-[(2-chloro-5-nitrobenzoyl)amino]-5-iodobenzoic acid
Mus musculus
pH 8.0, 37°C, recombinant enzyme
0.1
2-[(2-chloro-5-nitrobenzoyl)amino]-5-iodobenzoic acid
Mus musculus
above, pH 8.0, 37°C, recombinant enzyme
0.1
2-[(2-chloro-5-nitrobenzoyl)amino]-5-iodobenzoic acid
Rhipicephalus microplus
above, pH 8.0, 37°C, recombinant enzyme
0.0082
2-[(3-formyl-1H-indol-1-yl)methyl]benzonitrile
Ctenocephalides felis
pH 8.0, 37°C, recombinant enzyme
0.0089
2-[(3-formyl-1H-indol-1-yl)methyl]benzonitrile
Mus musculus
pH 8.0, 37°C, recombinant enzyme
0.0126
2-[(3-formyl-1H-indol-1-yl)methyl]benzonitrile
Mus musculus
pH 8.0, 37°C, recombinant enzyme
0.0138
2-[(3-formyl-1H-indol-1-yl)methyl]benzonitrile
Drosophila melanogaster
pH 8.0, 37°C, recombinant enzyme
0.014
2-[(3-formyl-1H-indol-1-yl)methyl]benzonitrile
Rhipicephalus microplus
pH 8.0, 37°C, recombinant enzyme
0.0002
3,3'-(4H-1,2,4-triazole-3,5-diyl)bis(4-nitro-1,2,5-oxadiazole)
Mus musculus
pH 8.0, 37°C, recombinant enzyme
0.0004
3,3'-(4H-1,2,4-triazole-3,5-diyl)bis(4-nitro-1,2,5-oxadiazole)
Mus musculus
pH 8.0, 37°C, recombinant enzyme
0.0148
3,3'-(4H-1,2,4-triazole-3,5-diyl)bis(4-nitro-1,2,5-oxadiazole)
Rhipicephalus microplus
pH 8.0, 37°C, recombinant enzyme
0.0196
3,3'-(4H-1,2,4-triazole-3,5-diyl)bis(4-nitro-1,2,5-oxadiazole)
Ctenocephalides felis
pH 8.0, 37°C, recombinant enzyme
0.0212
3,3'-(4H-1,2,4-triazole-3,5-diyl)bis(4-nitro-1,2,5-oxadiazole)
Drosophila melanogaster
pH 8.0, 37°C, recombinant enzyme
0.0123
3-Mercaptopropionic acid
Homo sapiens
-
-
0.0123
3-Mercaptopropionic acid
Homo sapiens
-
at 37°C
0.0123
3-Mercaptopropionic acid
Homo sapiens
-
at 37°C, pH not specified in the publication
0.0123
3-Mercaptopropionic acid
Homo sapiens
recombinant MBP-tagged enzyme, pH 8.0, 37°C
0.0202
3-[(2E)-2-[1-(3,4-dimethoxyphenyl)ethylidene]hydrazinyl]benzoic acid
Rhipicephalus microplus
pH 8.0, 37°C, recombinant enzyme
0.1
3-[(2E)-2-[1-(3,4-dimethoxyphenyl)ethylidene]hydrazinyl]benzoic acid
Mus musculus
above, pH 8.0, 37°C, recombinant enzyme
0.1
3-[(2E)-2-[1-(3,4-dimethoxyphenyl)ethylidene]hydrazinyl]benzoic acid
Ctenocephalides felis
above, pH 8.0, 37°C, recombinant enzyme
0.1
3-[(2E)-2-[1-(3,4-dimethoxyphenyl)ethylidene]hydrazinyl]benzoic acid
Drosophila melanogaster
above, pH 8.0, 37°C, recombinant enzyme
0.0063
3-[(E)-(2,6-difluorobenzylidene)amino]-2-thioxo-1,3-thiazolidin-4-one
Rhipicephalus microplus
pH 8.0, 37°C, recombinant enzyme
0.0064
3-[(E)-(2,6-difluorobenzylidene)amino]-2-thioxo-1,3-thiazolidin-4-one
Mus musculus
pH 8.0, 37°C, recombinant enzyme
0.0079
3-[(E)-(2,6-difluorobenzylidene)amino]-2-thioxo-1,3-thiazolidin-4-one
Mus musculus
pH 8.0, 37°C, recombinant enzyme
0.0109
3-[(E)-(2,6-difluorobenzylidene)amino]-2-thioxo-1,3-thiazolidin-4-one
Drosophila melanogaster
pH 8.0, 37°C, recombinant enzyme
0.0122
3-[(E)-(2,6-difluorobenzylidene)amino]-2-thioxo-1,3-thiazolidin-4-one
Ctenocephalides felis
pH 8.0, 37°C, recombinant enzyme
0.0072
4,4'-(phenylmethanediyl)bis[2-(4-chlorophenyl)-5-methyl-2,4-dihydro-3H-pyrazol-3-one]
Mus musculus
pH 8.0, 37°C, recombinant enzyme
0.012
4,4'-(phenylmethanediyl)bis[2-(4-chlorophenyl)-5-methyl-2,4-dihydro-3H-pyrazol-3-one]
Mus musculus
pH 8.0, 37°C, recombinant enzyme
0.0218
4,4'-(phenylmethanediyl)bis[2-(4-chlorophenyl)-5-methyl-2,4-dihydro-3H-pyrazol-3-one]
Ctenocephalides felis
pH 8.0, 37°C, recombinant enzyme
0.0269
4,4'-(phenylmethanediyl)bis[2-(4-chlorophenyl)-5-methyl-2,4-dihydro-3H-pyrazol-3-one]
Drosophila melanogaster
pH 8.0, 37°C, recombinant enzyme
0.099
4,4'-(phenylmethanediyl)bis[2-(4-chlorophenyl)-5-methyl-2,4-dihydro-3H-pyrazol-3-one]
Rhipicephalus microplus
pH 8.0, 37°C, recombinant enzyme
0.013
4,4'-[(4-hydroxyphenyl)methanediyl]bis(2-heptyl-5-methyl-2,4-dihydro-3H-pyrazol-3-one)
Mus musculus
pH 8.0, 37°C, recombinant enzyme
0.0138
4,4'-[(4-hydroxyphenyl)methanediyl]bis(2-heptyl-5-methyl-2,4-dihydro-3H-pyrazol-3-one)
Mus musculus
pH 8.0, 37°C, recombinant enzyme
0.0173
4,4'-[(4-hydroxyphenyl)methanediyl]bis(2-heptyl-5-methyl-2,4-dihydro-3H-pyrazol-3-one)
Ctenocephalides felis
pH 8.0, 37°C, recombinant enzyme
0.0188
4,4'-[(4-hydroxyphenyl)methanediyl]bis(2-heptyl-5-methyl-2,4-dihydro-3H-pyrazol-3-one)
Drosophila melanogaster
pH 8.0, 37°C, recombinant enzyme
0.0226
4,4'-[(4-hydroxyphenyl)methanediyl]bis(2-heptyl-5-methyl-2,4-dihydro-3H-pyrazol-3-one)
Rhipicephalus microplus
pH 8.0, 37°C, recombinant enzyme
0.0029
4-(morpholin-4-yl)naphthalene-1,2-dione
Mus musculus
pH 8.0, 37°C, recombinant enzyme
0.003
4-(morpholin-4-yl)naphthalene-1,2-dione
Drosophila melanogaster
pH 8.0, 37°C, recombinant enzyme
0.0034
4-(morpholin-4-yl)naphthalene-1,2-dione
Ctenocephalides felis
pH 8.0, 37°C, recombinant enzyme
0.0039
4-(morpholin-4-yl)naphthalene-1,2-dione
Rhipicephalus microplus
pH 8.0, 37°C, recombinant enzyme
0.0045
4-(morpholin-4-yl)naphthalene-1,2-dione
Mus musculus
pH 8.0, 37°C, recombinant enzyme
0.003
4-(piperidin-1-yl)naphthalene-1,2-dione
Drosophila melanogaster
pH 8.0, 37°C, recombinant enzyme
0.003
4-(piperidin-1-yl)naphthalene-1,2-dione
Mus musculus
pH 8.0, 37°C, recombinant enzyme
0.0038
4-(piperidin-1-yl)naphthalene-1,2-dione
Ctenocephalides felis
pH 8.0, 37°C, recombinant enzyme
0.0047
4-(piperidin-1-yl)naphthalene-1,2-dione
Mus musculus
pH 8.0, 37°C, recombinant enzyme
0.0053
4-(piperidin-1-yl)naphthalene-1,2-dione
Rhipicephalus microplus
pH 8.0, 37°C, recombinant enzyme
0.0034
4-nitro-1,6-dihydrobenzo[1,2-d:3,4-d']bis[1,2,3]triazole
Rhipicephalus microplus
pH 8.0, 37°C, recombinant enzyme
0.0077
4-nitro-1,6-dihydrobenzo[1,2-d:3,4-d']bis[1,2,3]triazole
Mus musculus
pH 8.0, 37°C, recombinant enzyme
0.0209
4-nitro-1,6-dihydrobenzo[1,2-d:3,4-d']bis[1,2,3]triazole
Drosophila melanogaster
pH 8.0, 37°C, recombinant enzyme
0.0211
4-nitro-1,6-dihydrobenzo[1,2-d:3,4-d']bis[1,2,3]triazole
Ctenocephalides felis
pH 8.0, 37°C, recombinant enzyme
0.065
4-nitro-1,6-dihydrobenzo[1,2-d:3,4-d']bis[1,2,3]triazole
Mus musculus
pH 8.0, 37°C, recombinant enzyme
0.0055
4-nitro-7-[[(1-phenyl-1H-tetrazol-5-yl)sulfanyl]methyl]-2,1,3-benzothiadiazole
Rhipicephalus microplus
pH 8.0, 37°C, recombinant enzyme
0.0912
4-nitro-7-[[(1-phenyl-1H-tetrazol-5-yl)sulfanyl]methyl]-2,1,3-benzothiadiazole
Ctenocephalides felis
pH 8.0, 37°C, recombinant enzyme
0.0981
4-nitro-7-[[(1-phenyl-1H-tetrazol-5-yl)sulfanyl]methyl]-2,1,3-benzothiadiazole
Drosophila melanogaster
pH 8.0, 37°C, recombinant enzyme
0.1
4-nitro-7-[[(1-phenyl-1H-tetrazol-5-yl)sulfanyl]methyl]-2,1,3-benzothiadiazole
Mus musculus
above, pH 8.0, 37°C, recombinant enzyme
0.0026
4-[(1,4-dioxo-1,2,3,4-tetrahydronaphthalen-2-yl)sulfanyl]butanoic acid
Rhipicephalus microplus
pH 8.0, 37°C, recombinant enzyme
0.0064
4-[(1,4-dioxo-1,2,3,4-tetrahydronaphthalen-2-yl)sulfanyl]butanoic acid
Mus musculus
pH 8.0, 37°C, recombinant enzyme
0.0067
4-[(1,4-dioxo-1,2,3,4-tetrahydronaphthalen-2-yl)sulfanyl]butanoic acid
Drosophila melanogaster
pH 8.0, 37°C, recombinant enzyme
0.0069
4-[(1,4-dioxo-1,2,3,4-tetrahydronaphthalen-2-yl)sulfanyl]butanoic acid
Ctenocephalides felis
pH 8.0, 37°C, recombinant enzyme
0.0112
4-[(1,4-dioxo-1,2,3,4-tetrahydronaphthalen-2-yl)sulfanyl]butanoic acid
Mus musculus
pH 8.0, 37°C, recombinant enzyme
0.0033
5,6-dichloro-2,1,3-benzothiadiazole-4,7-diol
Mus musculus
pH 8.0, 37°C, recombinant enzyme
0.0037
5,6-dichloro-2,1,3-benzothiadiazole-4,7-diol
Drosophila melanogaster
pH 8.0, 37°C, recombinant enzyme
0.0053
5,6-dichloro-2,1,3-benzothiadiazole-4,7-diol
Rhipicephalus microplus
pH 8.0, 37°C, recombinant enzyme
0.0057
5,6-dichloro-2,1,3-benzothiadiazole-4,7-diol
Ctenocephalides felis
pH 8.0, 37°C, recombinant enzyme
0.0083
5,6-dichloro-2,1,3-benzothiadiazole-4,7-diol
Mus musculus
pH 8.0, 37°C, recombinant enzyme
0.0069
5-[(E)-benzylideneamino]-6-[(2-hydroxyethyl)amino]pyrimidine-2,4(1H,3H)-dione
Mus musculus
pH 8.0, 37°C, recombinant enzyme
0.0077
5-[(E)-benzylideneamino]-6-[(2-hydroxyethyl)amino]pyrimidine-2,4(1H,3H)-dione
Drosophila melanogaster
pH 8.0, 37°C, recombinant enzyme
0.0087
5-[(E)-benzylideneamino]-6-[(2-hydroxyethyl)amino]pyrimidine-2,4(1H,3H)-dione
Ctenocephalides felis
pH 8.0, 37°C, recombinant enzyme
0.0104
5-[(E)-benzylideneamino]-6-[(2-hydroxyethyl)amino]pyrimidine-2,4(1H,3H)-dione
Mus musculus
pH 8.0, 37°C, recombinant enzyme
0.0104
5-[(E)-benzylideneamino]-6-[(2-hydroxyethyl)amino]pyrimidine-2,4(1H,3H)-dione
Rhipicephalus microplus
pH 8.0, 37°C, recombinant enzyme
0.0059
5-[(E)-[[1-(2-chlorobenzyl)-1H-indol-3-yl]methylidene]amino]-1,3-dihydro-2H-benzimidazol-2-one
Ctenocephalides felis
pH 8.0, 37°C, recombinant enzyme
0.0063
5-[(E)-[[1-(2-chlorobenzyl)-1H-indol-3-yl]methylidene]amino]-1,3-dihydro-2H-benzimidazol-2-one
Rhipicephalus microplus
pH 8.0, 37°C, recombinant enzyme
0.0065
5-[(E)-[[1-(2-chlorobenzyl)-1H-indol-3-yl]methylidene]amino]-1,3-dihydro-2H-benzimidazol-2-one
Mus musculus
pH 8.0, 37°C, recombinant enzyme
0.0066
5-[(E)-[[1-(2-chlorobenzyl)-1H-indol-3-yl]methylidene]amino]-1,3-dihydro-2H-benzimidazol-2-one
Drosophila melanogaster
pH 8.0, 37°C, recombinant enzyme
0.0129
5-[(E)-[[1-(2-chlorobenzyl)-1H-indol-3-yl]methylidene]amino]-1,3-dihydro-2H-benzimidazol-2-one
Mus musculus
pH 8.0, 37°C, recombinant enzyme
0.0122
5-[[5-hydroxy-3-methyl-1-(4-methylphenyl)-1H-pyrazol-4-yl]methylidene]-1,3-diphenyl-2-thioxodihydropyrimidine-4,6(1H,5H)-dione
Drosophila melanogaster
pH 8.0, 37°C, recombinant enzyme
0.0144
5-[[5-hydroxy-3-methyl-1-(4-methylphenyl)-1H-pyrazol-4-yl]methylidene]-1,3-diphenyl-2-thioxodihydropyrimidine-4,6(1H,5H)-dione
Ctenocephalides felis
pH 8.0, 37°C, recombinant enzyme
0.0149
5-[[5-hydroxy-3-methyl-1-(4-methylphenyl)-1H-pyrazol-4-yl]methylidene]-1,3-diphenyl-2-thioxodihydropyrimidine-4,6(1H,5H)-dione
Rhipicephalus microplus
pH 8.0, 37°C, recombinant enzyme
0.0558
5-[[5-hydroxy-3-methyl-1-(4-methylphenyl)-1H-pyrazol-4-yl]methylidene]-1,3-diphenyl-2-thioxodihydropyrimidine-4,6(1H,5H)-dione
Mus musculus
pH 8.0, 37°C, recombinant enzyme
0.0593
5-[[5-hydroxy-3-methyl-1-(4-methylphenyl)-1H-pyrazol-4-yl]methylidene]-1,3-diphenyl-2-thioxodihydropyrimidine-4,6(1H,5H)-dione
Mus musculus
pH 8.0, 37°C, recombinant enzyme
0.0021
6,11-dioxo-5a,6,11,11a-tetrahydronaphtho[2',3':4,5][1,3]thiazolo[3,2-a]pyridin-12-ium
Rhipicephalus microplus
pH 8.0, 37°C, recombinant enzyme
0.0022
6,11-dioxo-5a,6,11,11a-tetrahydronaphtho[2',3':4,5][1,3]thiazolo[3,2-a]pyridin-12-ium
Drosophila melanogaster
pH 8.0, 37°C, recombinant enzyme
0.0023
6,11-dioxo-5a,6,11,11a-tetrahydronaphtho[2',3':4,5][1,3]thiazolo[3,2-a]pyridin-12-ium
Mus musculus
pH 8.0, 37°C, recombinant enzyme
0.0029
6,11-dioxo-5a,6,11,11a-tetrahydronaphtho[2',3':4,5][1,3]thiazolo[3,2-a]pyridin-12-ium
Ctenocephalides felis
pH 8.0, 37°C, recombinant enzyme
0.0057
6,11-dioxo-5a,6,11,11a-tetrahydronaphtho[2',3':4,5][1,3]thiazolo[3,2-a]pyridin-12-ium
Mus musculus
pH 8.0, 37°C, recombinant enzyme
0.0045
9H-indeno[1,2-b][1,2,5]oxadiazolo[3,4-e]pyrazin-9-one
Rhipicephalus microplus
pH 8.0, 37°C, recombinant enzyme
0.0056
9H-indeno[1,2-b][1,2,5]oxadiazolo[3,4-e]pyrazin-9-one
Ctenocephalides felis
pH 8.0, 37°C, recombinant enzyme
0.0089
9H-indeno[1,2-b][1,2,5]oxadiazolo[3,4-e]pyrazin-9-one
Drosophila melanogaster
pH 8.0, 37°C, recombinant enzyme
0.0143
9H-indeno[1,2-b][1,2,5]oxadiazolo[3,4-e]pyrazin-9-one
Mus musculus
pH 8.0, 37°C, recombinant enzyme
0.1
9H-indeno[1,2-b][1,2,5]oxadiazolo[3,4-e]pyrazin-9-one
Mus musculus
above, pH 8.0, 37°C, recombinant enzyme
0.0049
biphenyl-3,3'-dicarbaldehyde
Mus musculus
pH 8.0, 37°C, recombinant enzyme
0.0053
biphenyl-3,3'-dicarbaldehyde
Rhipicephalus microplus
pH 8.0, 37°C, recombinant enzyme
0.0062
biphenyl-3,3'-dicarbaldehyde
Ctenocephalides felis
pH 8.0, 37°C, recombinant enzyme
0.0063
biphenyl-3,3'-dicarbaldehyde
Drosophila melanogaster
pH 8.0, 37°C, recombinant enzyme
0.0004
carboxymethoxylamine
Drosophila melanogaster
pH 8.0, 37°C, recombinant enzyme
0.0005
carboxymethoxylamine
Mus musculus
pH 8.0, 37°C, recombinant enzyme
0.001
carboxymethoxylamine
Mus musculus
pH 8.0, 37°C, recombinant enzyme
0.001
carboxymethoxylamine
Ctenocephalides felis
pH 8.0, 37°C, recombinant enzyme
0.001
methyl 2-amino-3-oxo-3H-phenothiazine-1-carboxylate
Mus musculus
pH 8.0, 37°C, recombinant enzyme
0.0014
methyl 2-amino-3-oxo-3H-phenothiazine-1-carboxylate
Drosophila melanogaster
pH 8.0, 37°C, recombinant enzyme
0.0015
methyl 2-amino-3-oxo-3H-phenothiazine-1-carboxylate
Ctenocephalides felis
pH 8.0, 37°C, recombinant enzyme
0.0017
methyl 2-amino-3-oxo-3H-phenothiazine-1-carboxylate
Rhipicephalus microplus
pH 8.0, 37°C, recombinant enzyme
0.002 - 4
methyl 2-amino-3-oxo-3H-phenothiazine-1-carboxylate
Mus musculus
pH 8.0, 37°C, recombinant enzyme
0.005
methyl 2-[[(2-methylimidazo[1,2-a]pyridin-3-yl)carbonyl]amino]benzoate
Drosophila melanogaster
pH 8.0, 37°C, recombinant enzyme
0.006
methyl 2-[[(2-methylimidazo[1,2-a]pyridin-3-yl)carbonyl]amino]benzoate
Rhipicephalus microplus
pH 8.0, 37°C, recombinant enzyme
0.0062
methyl 2-[[(2-methylimidazo[1,2-a]pyridin-3-yl)carbonyl]amino]benzoate
Ctenocephalides felis
pH 8.0, 37°C, recombinant enzyme
0.0065
methyl 2-[[(2-methylimidazo[1,2-a]pyridin-3-yl)carbonyl]amino]benzoate
Mus musculus
pH 8.0, 37°C, recombinant enzyme
0.0125
methyl 2-[[(2-methylimidazo[1,2-a]pyridin-3-yl)carbonyl]amino]benzoate
Mus musculus
pH 8.0, 37°C, recombinant enzyme
0.0076
N-(2-hydroxy-1,3-dioxo-2,3-dihydro-1H-inden-2-yl)benzamide
Mus musculus
pH 8.0, 37°C, recombinant enzyme
0.0082
N-(2-hydroxy-1,3-dioxo-2,3-dihydro-1H-inden-2-yl)benzamide
Rhipicephalus microplus
pH 8.0, 37°C, recombinant enzyme
0.0091
N-(2-hydroxy-1,3-dioxo-2,3-dihydro-1H-inden-2-yl)benzamide
Ctenocephalides felis
pH 8.0, 37°C, recombinant enzyme
0.0105
N-(2-hydroxy-1,3-dioxo-2,3-dihydro-1H-inden-2-yl)benzamide
Drosophila melanogaster
pH 8.0, 37°C, recombinant enzyme
0.0164
N-(2-hydroxy-1,3-dioxo-2,3-dihydro-1H-inden-2-yl)benzamide
Mus musculus
pH 8.0, 37°C, recombinant enzyme
0.001
N-[4,7-dioxo-6-(phenylamino)-4,7-dihydro-2,1,3-benzoxadiazol-5-yl]acetamide
Drosophila melanogaster
pH 8.0, 37°C, recombinant enzyme
0.0011
N-[4,7-dioxo-6-(phenylamino)-4,7-dihydro-2,1,3-benzoxadiazol-5-yl]acetamide
Ctenocephalides felis
pH 8.0, 37°C, recombinant enzyme
0.0011
N-[4,7-dioxo-6-(phenylamino)-4,7-dihydro-2,1,3-benzoxadiazol-5-yl]acetamide
Rhipicephalus microplus
pH 8.0, 37°C, recombinant enzyme
0.0012
N-[4,7-dioxo-6-(phenylamino)-4,7-dihydro-2,1,3-benzoxadiazol-5-yl]acetamide
Mus musculus
pH 8.0, 37°C, recombinant enzyme
0.0022
N-[4,7-dioxo-6-(phenylamino)-4,7-dihydro-2,1,3-benzoxadiazol-5-yl]acetamide
Mus musculus
pH 8.0, 37°C, recombinant enzyme
0.0013
N-[4,7-dioxo-6-(piperidin-1-yl)-4,7-dihydro-2,1,3-benzoxadiazol-5-yl]acetamide
Drosophila melanogaster
pH 8.0, 37°C, recombinant enzyme
0.0018
N-[4,7-dioxo-6-(piperidin-1-yl)-4,7-dihydro-2,1,3-benzoxadiazol-5-yl]acetamide
Ctenocephalides felis
pH 8.0, 37°C, recombinant enzyme
0.0022
N-[4,7-dioxo-6-(piperidin-1-yl)-4,7-dihydro-2,1,3-benzoxadiazol-5-yl]acetamide
Mus musculus
pH 8.0, 37°C, recombinant enzyme
0.0023
N-[4,7-dioxo-6-(piperidin-1-yl)-4,7-dihydro-2,1,3-benzoxadiazol-5-yl]acetamide
Rhipicephalus microplus
pH 8.0, 37°C, recombinant enzyme
0.0044
N-[4,7-dioxo-6-(piperidin-1-yl)-4,7-dihydro-2,1,3-benzoxadiazol-5-yl]acetamide
Mus musculus
pH 8.0, 37°C, recombinant enzyme
0.0037
naphtho[2',3':4,5]imidazo[1,2-a]pyridine-6,11-dione
Drosophila melanogaster
pH 8.0, 37°C, recombinant enzyme
0.0039
naphtho[2',3':4,5]imidazo[1,2-a]pyridine-6,11-dione
Ctenocephalides felis
pH 8.0, 37°C, recombinant enzyme
0.0041
naphtho[2',3':4,5]imidazo[1,2-a]pyridine-6,11-dione
Mus musculus
pH 8.0, 37°C, recombinant enzyme
0.0073
naphtho[2',3':4,5]imidazo[1,2-a]pyridine-6,11-dione
Rhipicephalus microplus
pH 8.0, 37°C, recombinant enzyme
0.0591
naphtho[2',3':4,5]imidazo[1,2-a]pyridine-6,11-dione
Mus musculus
pH 8.0, 37°C, recombinant enzyme
0.0244
[(1,3-dioxo-1,3-dihydro-2H-isoindol-2-yl)oxy]acetic acid
Drosophila melanogaster
pH 8.0, 37°C, recombinant enzyme
0.0257
[(1,3-dioxo-1,3-dihydro-2H-isoindol-2-yl)oxy]acetic acid
Ctenocephalides felis
pH 8.0, 37°C, recombinant enzyme
0.0284
[(1,3-dioxo-1,3-dihydro-2H-isoindol-2-yl)oxy]acetic acid
Rhipicephalus microplus
pH 8.0, 37°C, recombinant enzyme
0.1
[(1,3-dioxo-1,3-dihydro-2H-isoindol-2-yl)oxy]acetic acid
Mus musculus
above, pH 8.0, 37°C, recombinant enzyme