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3.4.24.63: meprin B

This is an abbreviated version!
For detailed information about meprin B, go to the full flat file.

Word Map on EC 3.4.24.63

Reaction

Hydrolysis of proteins, including azocasein, and peptides. Hydrolysis of -His5-/-Leu-, -Leu6-/-Cys-, -Ala14-/-Leu- and -Cys19-/-Gly- bonds in insulin B chain =

Synonyms

beta-secretase, cell surface sheddase, h-meprin beta, MEP1B, mephrin beta, meprin A subunit beta, Meprin b, meprin B metalloprotease, meprin beta, meprin beta metalloproteinase, meprin metalloprotease, meprin metalloproteinase, meprin metalloproteinase beta, meprin-beta, meprinbeta, metalloprotease meprin, metalloprotease meprin B, metalloprotease meprin beta, metalloproteinase meprin beta, Mmepb, More, mouse meprin beta, procollagen proteinase, Rmepb

ECTree

     3 Hydrolases
         3.4 Acting on peptide bonds (peptidases)
             3.4.24 Metalloendopeptidases
                3.4.24.63 meprin B

Turnover Number

Turnover Number on EC 3.4.24.63 - meprin B

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TURNOVER NUMBER [1/s]
SUBSTRATE
ORGANISM
UNIPROT
COMMENTARY hide
LITERATURE
IMAGE
71.7
Abz-MGWMDEIDK(Dnp)SG-OH
pH 8.0, 37°C, recombinant enzyme
13.5
Abz-VKMDAE-EDDnp
pH 7.5, 37°C
20.9
Abz-VNLDAE-EDDnp
pH 7.5, 37°C
35
Abz-YVAEAPK(Dnp)G-OH
pH 8.0, 37°C, recombinant enzyme
0.625
actin
-
pH 7.5, 37°C
15
alpha-MSH
-
pH 7.5, 37°C, mutant K185Y
11
bradykinin
-
pH 7.5, 37°C
13.9 - 15
cholecystokinin 8 sulfate
12.6
gastri-releasing peptide-(14-27)
-
pH 7.5, 37°C
12.4
gastrin
-
pH 7.5, 37°C
10.5 - 17.8
gastrin 17
15.9 - 26.8
glucagon
20
KKGYVADAP-4-nitroanilide
4
KKGYVADAP-7-amido-4-methylcoumarin
23.4
orcokinin
-
pH 7.5, 37°C
13.9
sCCK8NH2
-
pH 7.5, 37°C
150
villin
-
pH 7.5, 37°C
-