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0.001768
(1R,3S,4S,6R)-4-(2-carbamimidoylhydrazinyl)-6-guanidinocyclohexane-1,3-diyl bis(3-guanidinophenylcarbamate)
-
-
0.000812
(1R,3S,4S,6R)-4-(2-carbamimidoylhydrazinyl)-6-guanidinocyclohexane-1,3-diyl bis(4-guanidinophenylcarbamate)
-
-
0.00000099
(1S,14S,17S,20S,23S,26S,33r)-26-amino-N-(4-carbamimidoylbenzyl)-20,23-bis(3-guanidinopropyl)-17-neopentyl-4,8,16,19,22,25,32-heptaoxo-3,9,15,18,21,24,31-heptaazabicyclo[31.2.2]heptatriacontane-14-carboxamide
pH and temperature not specified in the publication
0.0000013
(D-Arg)9-amide
-
-
0.000046
1-[(1R,2R,4S,5S)-2,4-bis(4-carbamimidamidophenoxy)-5-[(4-carbamimidamidophenyl)amino]cyclohexyl]guanidine
-
-
0.000423
1-[4-([(1S,2S,4R,5R)-5-carbamimidamido-2,4-bis[(4-carbamimidamidonaphthalen-1-yl)oxy]cyclohexyl]amino)naphthalen-1-yl]guanidine
-
-
0.0000089
11-amino-undecanoyl-RARRRKKRT
-
pH 7.5, 37°C
0.000169
2-((1S,2S,4R,5R)-2,4-bis(2,4-diguanidinophenoxy)-5-guanidinocyclohexyl)hydrazinecarboximidamide
-
-
0.000404
2-((1S,2S,4R,5R)-2-(2,4-diguanidinophenoxy)-5-guanidino-4-(4-guanidinonaphthalen-1-yloxy)cyclohexyl)hydrazinecarboximidamide
-
-
0.000089
2-((1S,2S,4R,5R)-2-(2,4-diguanidinophenoxy)-5-guanidino-4-(4-guanidinophenoxy)cyclohexyl)hydrazinecarboximidamide
-
-
0.000022
2-((1S,2S,4R,5R)-2-(2-amino-4-guanidinophenoxy)-5-guanidino-4-(4-guanidinonaphthalen-1-yloxy)cyclohexyl)hydrazinecarboximidamide
-
-
0.000069
2-((1S,2S,4R,5R)-5-guanidino-2,4-bis(4-guanidinonaphthalen-1-yloxy)cyclohexyl)hydrazinecarboximidamide
-
-
0.000012
2-((1S,2S,4R,5R)-5-guanidino-2,4-bis(4-guanidinophenoxy)cyclohexyl)hydrazinecarboximidamide
-
-
0.000042
2-((1S,2S,4R,5R)-5-guanidino-2,4-bis(5-guanidinopyridin-2-yloxy)cyclohexyl)hydrazinecarboximidamide
-
-
0.000006
2-((1S,2S,4R,5R)-5-guanidino-4-(4-guanidinonaphthalen-1-yloxy)-2-(4-guanidinophenoxy)cyclohexyl)hydrazinecarboximidamide
-
-
0.012
2-(11-hydroxy-3-oxo-3H-dibenzo[c,h]xanthen-7-yl)benzoic acid
-
with CPA95 as substrate/with N-tert-butoxycarbonyl-Arg-Val-Arg-Arg-methylcoumarin amide as substrate
0.0033
3,3',3'',3'''-(1,4-phenylenebis(methanetriyl))tetrakis(4-hydroxy-2H-chromen-2-one)
-
with CPA95 as substrate
0.00104
3,3'-((2,3-dihydro-1H-inden-5-yl)methylene)bis(4-hydroxy-2H-chromen-2-one)
-
with CPA95 as substrate
0.1851
3,3'-((2-bromophenyl)methylene)bis(4-hydroxy-2H-chromen-2-one)
-
with Ac-Arg-Val-Arg-Arg-4-nitroanilide as substrate
0.0783
3,3'-((2-chlorophenyl)methylene)bis(4-hydroxy-2H-chromen-2-one)
-
with Ac-Arg-Val-Arg-Arg-4-nitroanilide as substrate
0.022
3,3'-((3,4,5-trimethoxyphenyl)methylene)bis(4-hydroxy-2H-chromen-2-one)
-
with Ac-Arg-Val-Arg-Arg-4-nitroanilide as substrate
0.0208
3,3'-((4-isopropoxyphenyl)methylene)bis(4-hydroxy-2H-chromen-2-one)
-
with Ac-Arg-Val-Arg-Arg-4-nitroanilide as substrate
0.00605
3,3'-(benzo[d][1,3]dioxol-5-ylmethylene)bis(4-hydroxy-2H-chromen-2-one)
-
with Ac-Arg-Val-Arg-Arg-4-nitroanilide as substrate
0.0188
3,3'-methylenebis(4-hydroxy-2H-chromen-2-one)
-
with CPA95 as substrate
2
3-(alpha-acetonyl-benzyl)-4-(hydroxycoumarin)
-
with Ac-Arg-Val-Arg-Arg-4-nitroanilide as substrate
0.0000025
3-guanidinomethylphenylacetyl-Val-Arg 4-amidinobenzylamide
pH 7.0, 22°C
0.0000000000224
4-aminomethyl-phenylacetyl-Arg-Tle-Arg-4-aminomethyl-benzamidine
pH and temperature not specified in the publication
1.3
4-hydroxy-3-oxo-1-phenylbutylcoumarin
-
with Ac-Arg-Val-Arg-Arg-4-nitroanilide as substrate
7.3
4-Hydroxycoumarin
-
with Ac-Arg-Val-Arg-Arg-4-nitroanilide as substrate
0.0000083
8-amino-octanoyl-RARRRKKRT
-
pH 7.5, 37°C
0.000019
Ac-Ac-RQIKIWFQNRRMKWKKRVR 4-amidinobenzylamide
pH and temperature not specified in the publication
0.0000228
Ac-AGYLLGKINLKALAALAKKILRVR 4-amidinobenzylamide
pH and temperature not specified in the publication
0.0024
Ac-D-Trp-D-Arg-D-Arg-D-Arg-D-Arg-D-Arg-NH2
-
pH 7.0, 37°C
0.0053
Ac-D-Trp-D-Arg-D-Arg-D-Arg-D-Arg-D-Leu-NH2
-
pH 7.0, 37°C
0.007
Ac-D-Trp-D-Arg-D-Arg-D-Arg-D-Ile-D-Arg-NH2
-
pH 7.0, 37°C
0.0227
Ac-D-Trp-D-Arg-D-Arg-D-Arg-D-Ile-D-Leu-NH2
-
pH 7.0, 37°C
0.0103
Ac-HHKRRR-NH2
-
pH 7.0, 37°C
0.0021
Ac-HRKRRR-NH2
-
pH 7.0, 37°C
0.0052
Ac-KHKRRR-NH2
-
pH 7.0, 37°C
0.0016
Ac-KRKRRR-NH2
-
pH 7.0, 37°C
0.0132
Ac-MHKRRR-NH2
-
pH 7.0, 37°C
0.0023
Ac-MRKRRR-NH2
-
pH 7.0, 37°C
0.0034
Ac-RHKRRR-NH2
-
pH 7.0, 37°C
0.0013
Ac-RRKRRR-NH2
-
pH 7.0, 37°C
0.0000107
Ac-RRRRRRRVR 4-amidinobenzylamide
pH and temperature not specified in the publication
0.000011
Ac-YGRKKRRQRRRVR 4-amidinobenzylamide
pH and temperature not specified in the publication
0.0000065
acetyl-RARRRKKRT
-
pH 7.5, 37°C
0.00239
acetyl-Val-Arg-4-amidinobenzylamide
-
pH 7.0, 37°C
0.0024
acetyl-Val-Arg-4-aminomethyl-benzamidine
pH and temperature not specified in the publication
0.0035
AcLLRVKR
-
pH 7.0, 37°C
0.0000094
Arg-Arg-Arg-Arg-Arg-Arg
pH and temperature not specified in the publication
0.000006
Arg-Arg-Arg-Arg-Arg-Arg-Arg-Arg
pH and temperature not specified in the publication
0.0000093
Arg-Arg-Arg-Arg-Arg-Arg-Arg-Arg-Arg-Arg
pH and temperature not specified in the publication
0.0000000754
Arg-Arg-Arg-Val-Arg 4-amidinobenzylamide
pH 7.0, 22°C
0.0000000337
Arg-Arg-Arg-Val-Arg-4-amidinobenzylamide
pH and temperature not specified in the publication
0.0000000000337
Arg-Arg-Arg-Val-Arg-4-aminomethyl-benzamidine
pH and temperature not specified in the publication
0.0000000119
Arg-Arg-Val-Arg 4-amidinobenzylamide
pH 7.0, 22°C
0.0000574
biotin-(8-(amino)-3,6-dioxa-octanoyl)2-Arg-Pro-Arg-4-amidinobenzylamide
-
pH 7.0, 37°C
0.000009
biotin-(8-(amino)-3,6-dioxa-octanoyl)2-Arg-Thr-Arg-4-amidinobenzylamide
-
pH 7.0, 37°C
0.0000151
biotin-(8-(amino)-3,6-dioxa-octanoyl)3-Arg-Pro-Arg-4-amidinobenzylamide
-
pH 7.0, 37°C
0.0000383
biotin-8-(amino)-3,6-dioxa-octanoyl-Arg-Pro-Arg-4-amidinobenzylamide
-
pH 7.0, 37°C
0.0042
biotin-8-(amino)-3,6-dioxa-octanoyl-Val-Arg-4-amidinobenzylamide
-
pH 7.0, 37°C
0.0000152
cholyl-RARRRKKRT
-
pH 7.5, 37°C
0.0000278
cyclo[(Arg)10]
pH and temperature not specified in the publication
0.0001104
cyclo[(Arg)6]
pH and temperature not specified in the publication
0.0000227
cyclo[(Arg)8]
pH and temperature not specified in the publication
0.00000068
cyclo[glutaryl-Arg-Arg-Arg-Lys]-Arg 4-amidinobenzylamide
pH and temperature not specified in the publication
0.000504
cyclo[glutaryl-Arg-Arg-Lys]-Arg 4-amidinobenzylamide
pH and temperature not specified in the publication
0.00000105
cyclo[glutaryl-Arg-Arg-Lys]-Lys 4-amidinobenzylamide
pH and temperature not specified in the publication
0.000000146
cyclo[succinyl-Phe-2-Nal-Arg-Arg-Arg-Arg-Arg-Lys]-Arg 4-amidinobenzylamide
pH and temperature not specified in the publication
0.000000154
cyclo[succinyl-Phe-2-Nal-Arg-Arg-Arg-Arg-Arg-Lys]-Lys 4-amidinobenzylamide
pH and temperature not specified in the publication
0.0000000538
cyclo[succinyl-Phe-2-Nal-Arg-Arg-Arg-Arg-Lys]-Arg 4-amidinobenzylamide
pH and temperature not specified in the publication
0.000000136
cyclo[succinyl-Phe-2-Nal-Arg-Arg-Arg-Arg-Lys]-Lys 4-amidinobenzylamide
pH and temperature not specified in the publication
0.000000378
cyclo[succinyl-Phe-2-Nal-Arg-Arg-Arg-Lys]-Arg 4-amidinobenzylamide
pH and temperature not specified in the publication
0.000000618
cyclo[succinyl-Phe-2-Nal-Arg-Arg-Arg-Lys]-Lys 4-amidinobenzylamide
pH and temperature not specified in the publication
0.0000000943
D-Arg-Arg-Arg-Val-Arg 4-amidinobenzylamide
pH 7.0, 22°C
0.000000491
D-Arg-Arg-Tle-Arg 4-amidinobenzylamide
pH 7.0, 22°C
0.0000000062
D-Arg-Arg-Val-Arg 4-amidinobenzylamide
pH 7.0, 22°C
0.000000108
D-Arg-D-Arg-Arg-Val-Arg 4-amidinobenzylamide
pH 7.0, 22°C
0.00000011
D-Arg-D-Arg-D-Arg-Arg-Val-Arg 4-amidinobenzylamide
pH 7.0, 22°C
0.0000000378
D-Arg-D-Arg-D-Arg-D-Arg-Arg-Val-Arg 4-amidinobenzylamide
pH 7.0, 22°C
0.0000078
eglin c mutant Arg replaced with Asp at P3
-
pH 7.5, 37°C
-
0.000023
eglin c mutant D42R, eglin c mutant L45R, eglin variant M1 RVTR
-
pH 7.5, 37°C
-
0.0000016
eglin variant M2 RVKR
-
pH 7.5, 37°C
-
0.00092
eglin variant M3 RVTRDERY
-
pH 7.5, 37°C
-
0.0003
eglin variant M4 RVTRDRRY
-
pH 7.5, 37°C
-
0.0000078
eglin variant M5 RVTRDLDY
-
pH 7.5, 37°C
-
0.000047
eglin variant M6 RVTRDLRR
-
pH 7.5, 37°C
-
0.000039
eglin variant M7 RVTRDLRE
-
pH 7.5, 37°C
-
0.00002
eglin variant M8 RVTRDARY
-
pH 7.5, 37°C
-
0.000068
hepta-L-arginine
-
pH 7.0, 37°C
0.000106
hexa-D-arginine
-
pH 7.0, 37°C
0.000156
hfurin25-107
-
pH 7.4, 37°C, versus N-benzyloxycarbonyl-RVRR-4-methylcoumarin 7-amide
-
0.0000000538
human proteinase inhibitor 8
-
pH 7.5, 37°C
-
0.00042
LLRVKR
-
pH 7.0, 37°C
0.0008 - 0.0034
LLRVKR-NH2
0.000000491
Lys-Arg-Arg-Tle-Lys 4-amidinobenzylamide (Lys1-Lys5 4-[4-(2-amino-2-oxoethyl)piperazin-1-yl]butanamide bridged)
pH and temperature not specified in the publication
0.00000504
Lys-Arg-Arg-Tle-Lys 4-amidinobenzylamide (Lys1-Lys5 N1-[[4-(2-amino-2-oxoethyl)phenyl]methyl]butanediamide bridged)
pH and temperature not specified in the publication
0.00000117
Lys-Arg-Arg-Tle-Lys 4-amidinobenzylamide (Lys1-Lys5 N1-[[4-(2-amino-2-oxoethyl)phenyl]methyl]pentanediamide bridged)
pH and temperature not specified in the publication
0.1452
methyl 4-(bis(4-hydroxy-2-oxo-2H-chromen-3-yl)methyl)benzoate
-
with Ac-Arg-Val-Arg-Arg-4-nitroanilide as substrate
0.0118
N''-[(1E)-[2-[(4-chlorobenzyl)oxy]phenyl]methylidene]carbonohydrazonic diamide
-
with Ac-Arg-Val-Arg-Arg-4-nitroanilide as substrate
0.00058
N-[3,5-bis[(1E)-1-(2-carbamimidoylhydrazinylidene)ethyl]phenyl]-2-[3-[(1E)-1-(2-carbamimidoylhydrazinylidene)ethyl]-5-[(1Z)-1-(2-carbamimidoylhydrazinylidene)ethyl]phenoxy]acetamide
-
pH 7.0,22°C
0.00046
N-[3,5-bis[(1E)-1-(2-carbamimidoylhydrazinylidene)ethyl]phenyl]-4-carbamimidamidobutanamide
-
pH 7.0,22°C
0.00104
N-[3,5-bis[(1E)-1-(2-carbamimidoylhydrazinylidene)ethyl]phenyl]-5-carbamimidamidopentanamide
-
pH 7.0,22°C
0.00113
N-[3,5-bis[(1E)-1-(2-carbamimidoylhydrazinylidene)ethyl]phenyl]-N'-[3-[(1E)-1-(2-carbamimidoylhydrazinylidene)ethyl]-5-[(1Z)-1-(2-carbamimidoylhydrazinylidene)ethyl]phenyl]propanediamide
-
pH 7.0,22°C
0.000000193
N2(carbamidoyl)Arg-Ala-Arg-Val-Arg 4-amidinobenzylamide
pH 7.0, 22°C
0.000000449
N2(carbamidoyl)Arg-Arg-Arg-Val-Arg 4-amidinobenzylamide
pH 7.0, 22°C
0.0002693
N2-(3-aminomethyl-phenylacetyl)-Val-Arg 4-amidinobenzylamide
pH 7.0, 22°C
0.0000000459
N2-(5-(guanidino)valeroyl)-Val-Arg 4-amidinobenzylamide
pH 7.0, 22°C
0.00000126 - 0.0000385
N2-(5-aminopentanoyl)-Val-Arg 4-amidinobenzylamide
0.0000267
N2-(5-guanidinopentanoly)-Val-Arg 4-amidinobenzylamide
pH 7.0, 22°C
0.00302
N2-(phenylacetyl)-L-arginyl-L-valyl-N-(3-aminopropyl)-L-argininamide
-
pH 7.0, temperature not specified in the publication
0.000063
N2-(phenylacetyl)-L-arginyl-L-valyl-N-(3-carbamimidamidopropyl)-L-argininamide
-
pH 7.0, temperature not specified in the publication
0.00749
N2-(phenylacetyl)-L-arginyl-L-valyl-N-(4-aminobutyl)-L-argininamide
-
pH 7.0, temperature not specified in the publication
0.000078
N2-(phenylacetyl)-L-arginyl-L-valyl-N-(4-carbamimidamidobutyl)-L-argininamide
-
pH 7.0, temperature not specified in the publication
0.00000081
N2-(phenylacetyl)-L-arginyl-L-valyl-N-(4-carbamimidoylbenzyl)-L-argininamide
-
pH 7.0, temperature not specified in the publication
0.000553
N2-(phenylacetyl)-L-arginyl-L-valyl-N-(5-aminopentyl)-L-argininamide
-
pH 7.0, temperature not specified in the publication
0.00107
N2-(phenylacetyl)-L-arginyl-L-valyl-N-(5-carbamimidamidopentyl)-L-argininamide
-
pH 7.0, temperature not specified in the publication
0.00971
N2-(phenylacetyl)-L-arginyl-L-valyl-N-(piperidin-4-ylmethyl)-L-argininamide
-
pH 7.0, temperature not specified in the publication
0.000053
N2-(phenylacetyl)-L-arginyl-L-valyl-N-[(1-carbamimidoylpiperidin-4-yl)methyl]-L-argininamide
-
pH 7.0, temperature not specified in the publication
0.00132
N2-(phenylacetyl)-L-arginyl-L-valyl-N-[3-(aminomethyl)benzyl]-L-argininamide
-
pH 7.0, temperature not specified in the publication
0.00273
N2-(phenylacetyl)-L-arginyl-L-valyl-N-[3-(carbamimidamidomethyl)benzyl]-L-argininamide
-
pH 7.0, temperature not specified in the publication
0.000627
N2-(phenylacetyl)-L-arginyl-L-valyl-N-[4-(aminomethyl)benzyl]-L-argininamide
-
pH 7.0, temperature not specified in the publication
0.00143
N2-(phenylacetyl)-L-arginyl-L-valyl-N-[4-(carbamimidamidomethyl)benzyl]-L-argininamide
-
pH 7.0, temperature not specified in the publication
0.0000000786
N2-acetyl-D-Leu-Leu-Leu-Leu-Arg-Val-Lys 4-amidinobenzylamide
pH 7.0, 22°C
0.000001
N2-acetyl-L-arginyl-L-valyl-N-(4-carbamimidoylbenzyl)-L-argininamide
-
pH 7.0, temperature not specified in the publication
0.000164
N2-acetyl-Leu-Leu-Leu-Leu-Arg-Tle-Arg 4-amidinobenzylamide
pH 7.0, 22°C
0.0000482
N2-acetyl-Leu-Leu-Leu-Leu-Arg-Tle-Lys 4-amidinobenzylamide
pH 7.0, 22°C
0.0000378
N2-acetyl-Leu-Leu-Leu-Leu-Arg-Val-Arg 4-amidinobenzylamide
pH 7.0, 22°C
0.000000164
N2-acetyl-Leu-Leu-Leu-Leu-Arg-Val-Lys 4-amidinobenzylamide
pH 7.0, 22°C
0.0000016
N2-decanoyl-L-arginyl-L-valyl-N-(4-carbamimidoylbenzyl)-L-argininamide
-
pH 7.0, temperature not specified in the publication
0.0000033
N2-decanoyl-L-arginyl-L-valyl-N-(4-carbamimidoylbenzyl)-L-lysinamide
-
pH 7.0, temperature not specified in the publication
0.000000051
N2-phenylacetyl-Ala-Arg-Arg-Val-Arg 4-amidinobenzylamide
pH 7.0, 22°C
0.0000000283
N2-phenylacetyl-Arg-Ala-Arg-Val-Arg 4-amidinobenzylamide
pH 7.0, 22°C
0.0000000337
N2-phenylacetyl-Arg-Arg-Arg-Val-Arg 4-amidinobenzylamide
pH 7.0, 22°C
0.0000000491
N2-phenylacetyl-Arg-Arg-Val-Arg 4-amidinobenzylamide
pH 7.0, 22°C
0.0000000563
N2-phenylacetyl-Arg-Val-Arg 4-amidinobenzylamide
pH 7.0, 22°C
0.0000000138
Nalpha(carbamidoyl)Arg-Arg-Val-Arg 4-amidinobenzylamide
pH 7.0, 22°C
0.00004 - 0.000042
nona-L-arginine
0.000061
octa-L-arginine
-
pH 7.0, 37°C
0.0193
PenLen (rSAAS-(221-246))
-
pH 7.4, 37°C
-
0.00099
penta-L-arginine
-
pH 7.0, 37°C
0.0000367
phenylacetyl-Arg-Pro-Arg-4-amidinobenzylamide
-
pH 7.0, 37°C
0.000006
phenylacetyl-Arg-Thr-Arg-4-amidinobenzylamide
-
pH 7.0, 37°C
0.00000081
phenylacetyl-Arg-Val-Arg-4-aminomethyl-benzamidine
pH and temperature not specified in the publication
0.000238
phenylacetyl-Cit-Arg-Val-Arg-4-aminomethyl-benzamidine
pH and temperature not specified in the publication
0.0009
profurin 39-62 DYYHFWHRGVKRSLSPHRPRHSR
-
pH 7.0, 25°C
0.0028
profurin 48-62 VTKRSLSPHRPRHSR
-
pH 7.0, 25°C
0.023
profurin 54-62 SPHRPRHSR
-
pH 7.0, 25°C
0.0007 - 0.0154
proPC1/3 39-62 NHYLF KHKSHPRRSALAITKR
0.0012
proPC1/3 39-62/A NAYLF KAKSAPRRSRRSALAITKR
-
pH 7.0, 25°C
0.0023
proPC1/3 50-62 RRSRR SALHITKR
-
pH 7.0, 25°C
0.0048
proPC1/3 50-83 RRSRRSALHITKRLSDDDRVTWAEQQYEKERSKR
-
pH 7.0, 25°C
0.0316
proPC1/3 55-62 SALHITKR
-
pH 7.0, 25°C
0.013
proPC1/3 55-62/A SALAITKR
-
pH 7.0, 25°C
0.0475
proPC1/3 74-83 QQYEKERSKR
-
pH 7.0, 25°C, competitive inhibition
0.000008
RARRRKKRT
-
pH 7.5, 37°C
0.000261
SAAS-(235-244)
-
pH 7.4, 37°C
0.0394
SAAS-(235-246)
-
pH 7.4, 37°C
-
0.00128
SAAS-(235-246)P1'A
-
pH 7.4, 37°
0.0044
SAAS-(235-246)P2'A
-
pH 7.4, 37°C
-
0.092
SAAS-(235-246)P3A
-
pH 7.4, 37°C
0.000114 - 0.0064
tetra-L-arginine
0.000038
TPQRARRRKKRF
-
-
0.000033
TPQRARRRKKRT
-
-
0.000034
TPQRARRRKKRW
-
-
0.000047
TPQRARRRKKRY
-
-
additional information
additional information
-
0.0008
LLRVKR-NH2
-
pH 7.0, 37°C
0.0034
LLRVKR-NH2
-
pH 7.0, 37°C
0.00000126
N2-(5-aminopentanoyl)-Val-Arg 4-amidinobenzylamide
pH 7.0, 22°C
0.0000385
N2-(5-aminopentanoyl)-Val-Arg 4-amidinobenzylamide
pH 7.0, 22°C
0.00004
nona-L-arginine
-
pH 7.0, 37°C
0.000042
nona-L-arginine
-
pH 7.0, 37°C
0.0007
proPC1/3 39-62 NHYLF KHKSHPRRSALAITKR
-
pH7.0, 25°C
0.0154
proPC1/3 39-62 NHYLF KHKSHPRRSALAITKR
-
pH 7.0, 25°C
0.000114
tetra-L-arginine
-
pH 7.0, 37°C
0.0064
tetra-L-arginine
-
pH 7.0, 37°C
0.000023
TPRARRRKKRT
-
-
0.000023
TPRARRRKKRT
-
pH 7.5, 37°C
additional information
additional information
-
inhibition kinetics
-
additional information
additional information
-
Ki-values of alpha1-antitrypsin and alpha1-antichymotrypsin mutants obtained by incorporation of furin recognition sequences within the reactive site loop of the molecule and modifying the P7-P1 region of the reactive site loop
-
additional information
additional information
Ki values of the inhibitors with inhibition constants above 0.1 nM are determined by fitting of the data to the equation for classical reversible competitive inhibition
-