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3.4.21.75: Furin

This is an abbreviated version!
For detailed information about Furin, go to the full flat file.

Word Map on EC 3.4.21.75

Reaction

Release of mature proteins from their proproteins by cleavage of -Arg-Xaa-Yaa-Arg-/- bonds, where Xaa can by any amino acid and Yaa is Arg or Lys. Releases albumin, complement component C3 and von Willebrand factor from their respective precursors =

Synonyms

Bfurin, Dfurin1, Dibasic processing enzyme, FUR, furin, furin A, furin B, furin convertase, furin protease, furin-like pro-protein convertase, furin-like prohormone convertase, furin-like proprotein convertase, furin-like protease, furin-like proteinase, FurinA, furinase, hfurin, KPC-1, More, PACE, Paired basic amino acid cleaving enzyme, Paired basic amino acid converting enzyme, Paired basic amino acid residue cleaving enzyme, PC1, PC1/3, PC2, PCSK3, proconvertase, prohormone convertase, prohormone convertase 1, prohormone convertase 2, Proprotein convertase, proprotein convertase subtilisin/kexin 3, proprotein convertase subtilisin/kexin type 3, proprotein convertase subtilisin/kexin type3, Serine proteinase PACE, Sfurin, sheddase, SPC3, subtilisin-like proprotein convertase, subtilisin-like protein convertase, Trans golgi network protease furin

ECTree

     3 Hydrolases
         3.4 Acting on peptide bonds (peptidases)
             3.4.21 Serine endopeptidases
                3.4.21.75 Furin

KI Value

KI Value on EC 3.4.21.75 - Furin

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Ki VALUE [mM]
INHIBITOR
ORGANISM
UNIPROT
COMMENTARY hide
LITERATURE
IMAGE
0.001768
(1R,3S,4S,6R)-4-(2-carbamimidoylhydrazinyl)-6-guanidinocyclohexane-1,3-diyl bis(3-guanidinophenylcarbamate)
-
-
0.000812
(1R,3S,4S,6R)-4-(2-carbamimidoylhydrazinyl)-6-guanidinocyclohexane-1,3-diyl bis(4-guanidinophenylcarbamate)
-
-
0.00000099
(1S,14S,17S,20S,23S,26S,33r)-26-amino-N-(4-carbamimidoylbenzyl)-20,23-bis(3-guanidinopropyl)-17-neopentyl-4,8,16,19,22,25,32-heptaoxo-3,9,15,18,21,24,31-heptaazabicyclo[31.2.2]heptatriacontane-14-carboxamide
pH and temperature not specified in the publication
0.0000013
(D-Arg)9-amide
-
-
0.000046
1-[(1R,2R,4S,5S)-2,4-bis(4-carbamimidamidophenoxy)-5-[(4-carbamimidamidophenyl)amino]cyclohexyl]guanidine
-
-
0.000423
1-[4-([(1S,2S,4R,5R)-5-carbamimidamido-2,4-bis[(4-carbamimidamidonaphthalen-1-yl)oxy]cyclohexyl]amino)naphthalen-1-yl]guanidine
-
-
0.0000089
11-amino-undecanoyl-RARRRKKRT
-
pH 7.5, 37°C
0.000169
2-((1S,2S,4R,5R)-2,4-bis(2,4-diguanidinophenoxy)-5-guanidinocyclohexyl)hydrazinecarboximidamide
-
-
0.000404
2-((1S,2S,4R,5R)-2-(2,4-diguanidinophenoxy)-5-guanidino-4-(4-guanidinonaphthalen-1-yloxy)cyclohexyl)hydrazinecarboximidamide
-
-
0.000089
2-((1S,2S,4R,5R)-2-(2,4-diguanidinophenoxy)-5-guanidino-4-(4-guanidinophenoxy)cyclohexyl)hydrazinecarboximidamide
-
-
0.000022
2-((1S,2S,4R,5R)-2-(2-amino-4-guanidinophenoxy)-5-guanidino-4-(4-guanidinonaphthalen-1-yloxy)cyclohexyl)hydrazinecarboximidamide
-
-
0.000069
2-((1S,2S,4R,5R)-5-guanidino-2,4-bis(4-guanidinonaphthalen-1-yloxy)cyclohexyl)hydrazinecarboximidamide
-
-
0.000012
2-((1S,2S,4R,5R)-5-guanidino-2,4-bis(4-guanidinophenoxy)cyclohexyl)hydrazinecarboximidamide
-
-
0.000042
2-((1S,2S,4R,5R)-5-guanidino-2,4-bis(5-guanidinopyridin-2-yloxy)cyclohexyl)hydrazinecarboximidamide
-
-
0.000006
2-((1S,2S,4R,5R)-5-guanidino-4-(4-guanidinonaphthalen-1-yloxy)-2-(4-guanidinophenoxy)cyclohexyl)hydrazinecarboximidamide
-
-
0.012
2-(11-hydroxy-3-oxo-3H-dibenzo[c,h]xanthen-7-yl)benzoic acid
-
with CPA95 as substrate/with N-tert-butoxycarbonyl-Arg-Val-Arg-Arg-methylcoumarin amide as substrate
0.0033
3,3',3'',3'''-(1,4-phenylenebis(methanetriyl))tetrakis(4-hydroxy-2H-chromen-2-one)
-
with CPA95 as substrate
0.00104
3,3'-((2,3-dihydro-1H-inden-5-yl)methylene)bis(4-hydroxy-2H-chromen-2-one)
-
with CPA95 as substrate
0.1851
3,3'-((2-bromophenyl)methylene)bis(4-hydroxy-2H-chromen-2-one)
-
with Ac-Arg-Val-Arg-Arg-4-nitroanilide as substrate
0.0783
3,3'-((2-chlorophenyl)methylene)bis(4-hydroxy-2H-chromen-2-one)
-
with Ac-Arg-Val-Arg-Arg-4-nitroanilide as substrate
0.022
3,3'-((3,4,5-trimethoxyphenyl)methylene)bis(4-hydroxy-2H-chromen-2-one)
-
with Ac-Arg-Val-Arg-Arg-4-nitroanilide as substrate
0.0208
3,3'-((4-isopropoxyphenyl)methylene)bis(4-hydroxy-2H-chromen-2-one)
-
with Ac-Arg-Val-Arg-Arg-4-nitroanilide as substrate
0.00605
3,3'-(benzo[d][1,3]dioxol-5-ylmethylene)bis(4-hydroxy-2H-chromen-2-one)
-
with Ac-Arg-Val-Arg-Arg-4-nitroanilide as substrate
0.0188
3,3'-methylenebis(4-hydroxy-2H-chromen-2-one)
-
with CPA95 as substrate
2
3-(alpha-acetonyl-benzyl)-4-(hydroxycoumarin)
-
with Ac-Arg-Val-Arg-Arg-4-nitroanilide as substrate
0.0000025
3-guanidinomethylphenylacetyl-Val-Arg 4-amidinobenzylamide
pH 7.0, 22°C
0.0000000000224
4-aminomethyl-phenylacetyl-Arg-Tle-Arg-4-aminomethyl-benzamidine
pH and temperature not specified in the publication
1.3
4-hydroxy-3-oxo-1-phenylbutylcoumarin
-
with Ac-Arg-Val-Arg-Arg-4-nitroanilide as substrate
7.3
4-Hydroxycoumarin
-
with Ac-Arg-Val-Arg-Arg-4-nitroanilide as substrate
0.0000083
8-amino-octanoyl-RARRRKKRT
-
pH 7.5, 37°C
0.000019
Ac-Ac-RQIKIWFQNRRMKWKKRVR 4-amidinobenzylamide
pH and temperature not specified in the publication
0.0000228
Ac-AGYLLGKINLKALAALAKKILRVR 4-amidinobenzylamide
pH and temperature not specified in the publication
0.0024
Ac-D-Trp-D-Arg-D-Arg-D-Arg-D-Arg-D-Arg-NH2
-
pH 7.0, 37°C
0.0053
Ac-D-Trp-D-Arg-D-Arg-D-Arg-D-Arg-D-Leu-NH2
-
pH 7.0, 37°C
0.007
Ac-D-Trp-D-Arg-D-Arg-D-Arg-D-Ile-D-Arg-NH2
-
pH 7.0, 37°C
0.0227
Ac-D-Trp-D-Arg-D-Arg-D-Arg-D-Ile-D-Leu-NH2
-
pH 7.0, 37°C
0.0103
Ac-HHKRRR-NH2
-
pH 7.0, 37°C
0.0021
Ac-HRKRRR-NH2
-
pH 7.0, 37°C
0.0052
Ac-KHKRRR-NH2
-
pH 7.0, 37°C
0.0016
Ac-KRKRRR-NH2
-
pH 7.0, 37°C
0.0132
Ac-MHKRRR-NH2
-
pH 7.0, 37°C
0.0023
Ac-MRKRRR-NH2
-
pH 7.0, 37°C
0.0034
Ac-RHKRRR-NH2
-
pH 7.0, 37°C
0.0013
Ac-RRKRRR-NH2
-
pH 7.0, 37°C
0.0000107
Ac-RRRRRRRVR 4-amidinobenzylamide
pH and temperature not specified in the publication
0.000011
Ac-YGRKKRRQRRRVR 4-amidinobenzylamide
pH and temperature not specified in the publication
0.0000065
acetyl-RARRRKKRT
-
pH 7.5, 37°C
0.00239
acetyl-Val-Arg-4-amidinobenzylamide
-
pH 7.0, 37°C
0.0024
acetyl-Val-Arg-4-aminomethyl-benzamidine
pH and temperature not specified in the publication
0.0035
AcLLRVKR
-
pH 7.0, 37°C
0.0000094
Arg-Arg-Arg-Arg-Arg-Arg
pH and temperature not specified in the publication
0.000006
Arg-Arg-Arg-Arg-Arg-Arg-Arg-Arg
pH and temperature not specified in the publication
0.0000093
Arg-Arg-Arg-Arg-Arg-Arg-Arg-Arg-Arg-Arg
pH and temperature not specified in the publication
0.0000000754
Arg-Arg-Arg-Val-Arg 4-amidinobenzylamide
pH 7.0, 22°C
0.0000000337
Arg-Arg-Arg-Val-Arg-4-amidinobenzylamide
pH and temperature not specified in the publication
0.0000000000337
Arg-Arg-Arg-Val-Arg-4-aminomethyl-benzamidine
pH and temperature not specified in the publication
0.0000000119
Arg-Arg-Val-Arg 4-amidinobenzylamide
pH 7.0, 22°C
0.0000574
biotin-(8-(amino)-3,6-dioxa-octanoyl)2-Arg-Pro-Arg-4-amidinobenzylamide
-
pH 7.0, 37°C
0.000009
biotin-(8-(amino)-3,6-dioxa-octanoyl)2-Arg-Thr-Arg-4-amidinobenzylamide
-
pH 7.0, 37°C
0.0000151
biotin-(8-(amino)-3,6-dioxa-octanoyl)3-Arg-Pro-Arg-4-amidinobenzylamide
-
pH 7.0, 37°C
0.0000383
biotin-8-(amino)-3,6-dioxa-octanoyl-Arg-Pro-Arg-4-amidinobenzylamide
-
pH 7.0, 37°C
0.0042
biotin-8-(amino)-3,6-dioxa-octanoyl-Val-Arg-4-amidinobenzylamide
-
pH 7.0, 37°C
0.0000152
cholyl-RARRRKKRT
-
pH 7.5, 37°C
0.0000278
cyclo[(Arg)10]
pH and temperature not specified in the publication
0.0001104
cyclo[(Arg)6]
pH and temperature not specified in the publication
0.0000227
cyclo[(Arg)8]
pH and temperature not specified in the publication
0.00000068
cyclo[glutaryl-Arg-Arg-Arg-Lys]-Arg 4-amidinobenzylamide
pH and temperature not specified in the publication
0.000504
cyclo[glutaryl-Arg-Arg-Lys]-Arg 4-amidinobenzylamide
pH and temperature not specified in the publication
0.00000105
cyclo[glutaryl-Arg-Arg-Lys]-Lys 4-amidinobenzylamide
pH and temperature not specified in the publication
0.000000146
cyclo[succinyl-Phe-2-Nal-Arg-Arg-Arg-Arg-Arg-Lys]-Arg 4-amidinobenzylamide
pH and temperature not specified in the publication
0.000000154
cyclo[succinyl-Phe-2-Nal-Arg-Arg-Arg-Arg-Arg-Lys]-Lys 4-amidinobenzylamide
pH and temperature not specified in the publication
0.0000000538
cyclo[succinyl-Phe-2-Nal-Arg-Arg-Arg-Arg-Lys]-Arg 4-amidinobenzylamide
pH and temperature not specified in the publication
0.000000136
cyclo[succinyl-Phe-2-Nal-Arg-Arg-Arg-Arg-Lys]-Lys 4-amidinobenzylamide
pH and temperature not specified in the publication
0.000000378
cyclo[succinyl-Phe-2-Nal-Arg-Arg-Arg-Lys]-Arg 4-amidinobenzylamide
pH and temperature not specified in the publication
0.000000618
cyclo[succinyl-Phe-2-Nal-Arg-Arg-Arg-Lys]-Lys 4-amidinobenzylamide
pH and temperature not specified in the publication
0.0000000943
D-Arg-Arg-Arg-Val-Arg 4-amidinobenzylamide
pH 7.0, 22°C
0.000000491
D-Arg-Arg-Tle-Arg 4-amidinobenzylamide
pH 7.0, 22°C
0.0000000062
D-Arg-Arg-Val-Arg 4-amidinobenzylamide
pH 7.0, 22°C
0.000000108
D-Arg-D-Arg-Arg-Val-Arg 4-amidinobenzylamide
pH 7.0, 22°C
0.00000011
D-Arg-D-Arg-D-Arg-Arg-Val-Arg 4-amidinobenzylamide
pH 7.0, 22°C
0.0000000378
D-Arg-D-Arg-D-Arg-D-Arg-Arg-Val-Arg 4-amidinobenzylamide
pH 7.0, 22°C
0.0000078
eglin c mutant Arg replaced with Asp at P3
-
pH 7.5, 37°C
-
0.000023
eglin c mutant D42R, eglin c mutant L45R, eglin variant M1 RVTR
-
pH 7.5, 37°C
-
0.0000016
eglin variant M2 RVKR
-
pH 7.5, 37°C
-
0.00092
eglin variant M3 RVTRDERY
-
pH 7.5, 37°C
-
0.0003
eglin variant M4 RVTRDRRY
-
pH 7.5, 37°C
-
0.0000078
eglin variant M5 RVTRDLDY
-
pH 7.5, 37°C
-
0.000047
eglin variant M6 RVTRDLRR
-
pH 7.5, 37°C
-
0.000039
eglin variant M7 RVTRDLRE
-
pH 7.5, 37°C
-
0.00002
eglin variant M8 RVTRDARY
-
pH 7.5, 37°C
-
0.000068
hepta-L-arginine
-
pH 7.0, 37°C
0.000106
hexa-D-arginine
-
pH 7.0, 37°C
0.000156
hfurin25-107
-
pH 7.4, 37°C, versus N-benzyloxycarbonyl-RVRR-4-methylcoumarin 7-amide
-
0.0000000538
human proteinase inhibitor 8
-
pH 7.5, 37°C
-
0.00042
LLRVKR
-
pH 7.0, 37°C
0.0008 - 0.0034
LLRVKR-NH2
0.000000491
Lys-Arg-Arg-Tle-Lys 4-amidinobenzylamide (Lys1-Lys5 4-[4-(2-amino-2-oxoethyl)piperazin-1-yl]butanamide bridged)
pH and temperature not specified in the publication
0.00000504
Lys-Arg-Arg-Tle-Lys 4-amidinobenzylamide (Lys1-Lys5 N1-[[4-(2-amino-2-oxoethyl)phenyl]methyl]butanediamide bridged)
pH and temperature not specified in the publication
0.00000117
Lys-Arg-Arg-Tle-Lys 4-amidinobenzylamide (Lys1-Lys5 N1-[[4-(2-amino-2-oxoethyl)phenyl]methyl]pentanediamide bridged)
pH and temperature not specified in the publication
0.1452
methyl 4-(bis(4-hydroxy-2-oxo-2H-chromen-3-yl)methyl)benzoate
-
with Ac-Arg-Val-Arg-Arg-4-nitroanilide as substrate
0.0118
N''-[(1E)-[2-[(4-chlorobenzyl)oxy]phenyl]methylidene]carbonohydrazonic diamide
-
with Ac-Arg-Val-Arg-Arg-4-nitroanilide as substrate
0.00058
N-[3,5-bis[(1E)-1-(2-carbamimidoylhydrazinylidene)ethyl]phenyl]-2-[3-[(1E)-1-(2-carbamimidoylhydrazinylidene)ethyl]-5-[(1Z)-1-(2-carbamimidoylhydrazinylidene)ethyl]phenoxy]acetamide
-
pH 7.0,22°C
0.00046
N-[3,5-bis[(1E)-1-(2-carbamimidoylhydrazinylidene)ethyl]phenyl]-4-carbamimidamidobutanamide
-
pH 7.0,22°C
0.00104
N-[3,5-bis[(1E)-1-(2-carbamimidoylhydrazinylidene)ethyl]phenyl]-5-carbamimidamidopentanamide
-
pH 7.0,22°C
0.00113
N-[3,5-bis[(1E)-1-(2-carbamimidoylhydrazinylidene)ethyl]phenyl]-N'-[3-[(1E)-1-(2-carbamimidoylhydrazinylidene)ethyl]-5-[(1Z)-1-(2-carbamimidoylhydrazinylidene)ethyl]phenyl]propanediamide
-
pH 7.0,22°C
0.000000193
N2(carbamidoyl)Arg-Ala-Arg-Val-Arg 4-amidinobenzylamide
pH 7.0, 22°C
0.000000449
N2(carbamidoyl)Arg-Arg-Arg-Val-Arg 4-amidinobenzylamide
pH 7.0, 22°C
0.0002693
N2-(3-aminomethyl-phenylacetyl)-Val-Arg 4-amidinobenzylamide
pH 7.0, 22°C
0.0000000459
N2-(5-(guanidino)valeroyl)-Val-Arg 4-amidinobenzylamide
pH 7.0, 22°C
0.00000126 - 0.0000385
N2-(5-aminopentanoyl)-Val-Arg 4-amidinobenzylamide
0.0000267
N2-(5-guanidinopentanoly)-Val-Arg 4-amidinobenzylamide
pH 7.0, 22°C
0.00302
N2-(phenylacetyl)-L-arginyl-L-valyl-N-(3-aminopropyl)-L-argininamide
-
pH 7.0, temperature not specified in the publication
0.000063
N2-(phenylacetyl)-L-arginyl-L-valyl-N-(3-carbamimidamidopropyl)-L-argininamide
-
pH 7.0, temperature not specified in the publication
0.00749
N2-(phenylacetyl)-L-arginyl-L-valyl-N-(4-aminobutyl)-L-argininamide
-
pH 7.0, temperature not specified in the publication
0.000078
N2-(phenylacetyl)-L-arginyl-L-valyl-N-(4-carbamimidamidobutyl)-L-argininamide
-
pH 7.0, temperature not specified in the publication
0.00000081
N2-(phenylacetyl)-L-arginyl-L-valyl-N-(4-carbamimidoylbenzyl)-L-argininamide
-
pH 7.0, temperature not specified in the publication
0.000553
N2-(phenylacetyl)-L-arginyl-L-valyl-N-(5-aminopentyl)-L-argininamide
-
pH 7.0, temperature not specified in the publication
0.00107
N2-(phenylacetyl)-L-arginyl-L-valyl-N-(5-carbamimidamidopentyl)-L-argininamide
-
pH 7.0, temperature not specified in the publication
0.00971
N2-(phenylacetyl)-L-arginyl-L-valyl-N-(piperidin-4-ylmethyl)-L-argininamide
-
pH 7.0, temperature not specified in the publication
0.000053
N2-(phenylacetyl)-L-arginyl-L-valyl-N-[(1-carbamimidoylpiperidin-4-yl)methyl]-L-argininamide
-
pH 7.0, temperature not specified in the publication
0.00132
N2-(phenylacetyl)-L-arginyl-L-valyl-N-[3-(aminomethyl)benzyl]-L-argininamide
-
pH 7.0, temperature not specified in the publication
0.00273
N2-(phenylacetyl)-L-arginyl-L-valyl-N-[3-(carbamimidamidomethyl)benzyl]-L-argininamide
-
pH 7.0, temperature not specified in the publication
0.000627
N2-(phenylacetyl)-L-arginyl-L-valyl-N-[4-(aminomethyl)benzyl]-L-argininamide
-
pH 7.0, temperature not specified in the publication
0.00143
N2-(phenylacetyl)-L-arginyl-L-valyl-N-[4-(carbamimidamidomethyl)benzyl]-L-argininamide
-
pH 7.0, temperature not specified in the publication
0.0000000786
N2-acetyl-D-Leu-Leu-Leu-Leu-Arg-Val-Lys 4-amidinobenzylamide
pH 7.0, 22°C
0.000001
N2-acetyl-L-arginyl-L-valyl-N-(4-carbamimidoylbenzyl)-L-argininamide
-
pH 7.0, temperature not specified in the publication
0.000164
N2-acetyl-Leu-Leu-Leu-Leu-Arg-Tle-Arg 4-amidinobenzylamide
pH 7.0, 22°C
0.0000482
N2-acetyl-Leu-Leu-Leu-Leu-Arg-Tle-Lys 4-amidinobenzylamide
pH 7.0, 22°C
0.0000378
N2-acetyl-Leu-Leu-Leu-Leu-Arg-Val-Arg 4-amidinobenzylamide
pH 7.0, 22°C
0.000000164
N2-acetyl-Leu-Leu-Leu-Leu-Arg-Val-Lys 4-amidinobenzylamide
pH 7.0, 22°C
0.0000016
N2-decanoyl-L-arginyl-L-valyl-N-(4-carbamimidoylbenzyl)-L-argininamide
-
pH 7.0, temperature not specified in the publication
0.0000033
N2-decanoyl-L-arginyl-L-valyl-N-(4-carbamimidoylbenzyl)-L-lysinamide
-
pH 7.0, temperature not specified in the publication
0.000000051
N2-phenylacetyl-Ala-Arg-Arg-Val-Arg 4-amidinobenzylamide
pH 7.0, 22°C
0.0000000283
N2-phenylacetyl-Arg-Ala-Arg-Val-Arg 4-amidinobenzylamide
pH 7.0, 22°C
0.0000000337
N2-phenylacetyl-Arg-Arg-Arg-Val-Arg 4-amidinobenzylamide
pH 7.0, 22°C
0.0000000491
N2-phenylacetyl-Arg-Arg-Val-Arg 4-amidinobenzylamide
pH 7.0, 22°C
0.0000000563
N2-phenylacetyl-Arg-Val-Arg 4-amidinobenzylamide
pH 7.0, 22°C
0.0000000138
Nalpha(carbamidoyl)Arg-Arg-Val-Arg 4-amidinobenzylamide
pH 7.0, 22°C
0.00004 - 0.000042
nona-L-arginine
0.000061
octa-L-arginine
-
pH 7.0, 37°C
0.0193
PenLen (rSAAS-(221-246))
-
pH 7.4, 37°C
-
0.00099
penta-L-arginine
-
pH 7.0, 37°C
0.0000367
phenylacetyl-Arg-Pro-Arg-4-amidinobenzylamide
-
pH 7.0, 37°C
0.000006
phenylacetyl-Arg-Thr-Arg-4-amidinobenzylamide
-
pH 7.0, 37°C
0.00000081
phenylacetyl-Arg-Val-Arg-4-aminomethyl-benzamidine
pH and temperature not specified in the publication
0.000238
phenylacetyl-Cit-Arg-Val-Arg-4-aminomethyl-benzamidine
pH and temperature not specified in the publication
0.0009
profurin 39-62 DYYHFWHRGVKRSLSPHRPRHSR
-
pH 7.0, 25°C
0.0028
profurin 48-62 VTKRSLSPHRPRHSR
-
pH 7.0, 25°C
0.023
profurin 54-62 SPHRPRHSR
-
pH 7.0, 25°C
0.0007 - 0.0154
proPC1/3 39-62 NHYLF KHKSHPRRSALAITKR
0.0012
proPC1/3 39-62/A NAYLF KAKSAPRRSRRSALAITKR
-
pH 7.0, 25°C
0.0023
proPC1/3 50-62 RRSRR SALHITKR
-
pH 7.0, 25°C
0.0048
proPC1/3 50-83 RRSRRSALHITKRLSDDDRVTWAEQQYEKERSKR
-
pH 7.0, 25°C
0.0316
proPC1/3 55-62 SALHITKR
-
pH 7.0, 25°C
0.013
proPC1/3 55-62/A SALAITKR
-
pH 7.0, 25°C
0.0475
proPC1/3 74-83 QQYEKERSKR
-
pH 7.0, 25°C, competitive inhibition
0.000008
RARRRKKRT
-
pH 7.5, 37°C
0.000261
SAAS-(235-244)
-
pH 7.4, 37°C
0.0394
SAAS-(235-246)
-
pH 7.4, 37°C
-
0.00128
SAAS-(235-246)P1'A
-
pH 7.4, 37°
0.0044
SAAS-(235-246)P2'A
-
pH 7.4, 37°C
-
0.092
SAAS-(235-246)P3A
-
pH 7.4, 37°C
0.000114 - 0.0064
tetra-L-arginine
0.000038
TPQRARRRKKRF
-
-
0.000033
TPQRARRRKKRT
-
-
0.000034
TPQRARRRKKRW
-
-
0.000047
TPQRARRRKKRY
-
-
0.000057
TPRARRRKKRG
-
-
0.00003
TPRARRRKKRI
-
-
0.000023
TPRARRRKKRT
additional information
additional information
-