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0.93 - 19.3
Ala-Ala-Pro-Leu-4-nitroanilide
0.098 - 23
Ala-Ala-Pro-Met-4-nitroanilide
0.028 - 143
Ala-Ala-Pro-Phe-4-nitroanilide
24.7 - 25.6
Big endothelin-1
13
H2N(CH2)5CO-Ala-Ala-Pro-Phe-4-nitroanilide
-
-
10
methoxysuccinyl-Ala-Ala-Pro-Phe-4-nitroanilide
-
-
6.7
succinyl-Ala-Ala-Pro-Leu-4-nitroanilide
-
-
2.5
succinyl-Ala-Ala-Pro-Met-4-nitroanilide
-
-
1.25 - 65
succinyl-Ala-Ala-Pro-Phe-4-nitroanilide
38 - 51
succinyl-Ala-Pro-Phe-4-nitroanilide
17
succinyl-Ala-Val-Pro-Phe-4-nitroanilide
-
-
4.7
succinyl-epsilon-(2-picolinyl)Lys-Pro-Phe-4-nitroanilide
-
-
86 - 480
succinyl-epsilon-(2-picolinyl)Lys-Val-Pro-Phe-4-nitroanilide
56 - 86
succinyl-Gln-Pro-Phe-4-nitroanilide
9.2 - 61
succinyl-Glu-Pro-Phe-4-nitroanilide
53 - 68
succinyl-Glu-Val-Pro-Phe-4-nitroanilide
2.5 - 3.6
succinyl-L-Ala-L-Ala-L-Pro-L-Phe-4-nitroanilide
12.6 - 17.8
succinyl-L-Ala-L-Ala-L-Pro-L-Phe-thiobenzyl ester
37 - 77
succinyl-Leu-Pro-Phe-4-nitroanilide
19 - 79
succinyl-Leu-Val-Pro-Phe-4-nitroanilide
14 - 32
succinyl-Lys-Pro-Phe-4-nitroanilide
58 - 66
succinyl-Lys-Val-Pro-Phe-4-nitroanilide
25 - 100
succinyl-Met-Pro-Phe-4-nitroanilide
25 - 53
succinyl-Met-Val-Pro-Phe-4-nitroanilide
7.1 - 10
succinyl-Phe-Ala-Phe-4-nitroanilide
23
succinyl-Phe-epsilon-(2-picolinyl)Lys-4-nitroanilide
-
-
3.9 - 25
succinyl-Phe-Gln-Phe-4-nitroanilide
0.9 - 8.4
succinyl-Phe-Glu-Phe-4-nitroanilide
7.5 - 19
succinyl-Phe-Leu-Phe-4-nitroanilide
18
succinyl-Phe-Lys-Phe-4-nitroanilide
-
-
5.9 - 8.2
succinyl-Phe-Met-Phe-4-nitroanilide
17 - 28
succinyl-Phe-Pro-Phe-4-nitroanilide
11 - 19
succinyl-Phe-Pro-Thr-Phe-4-nitroanilide
5.4 - 6.2
succinyl-Phe-Ser-Phe-4-nitroanilide
9.3 - 10
succinyl-Phe-Thr-Phe-4-nitroanilide
4 - 15
succinyl-Phe-Val-Phe-4-nitroanilide
24 - 56
succinyl-Phe-Val-Pro-Phe-4-nitroanilide
20 - 38
succinyl-Ser-Pro-Phe-4-nitroanilide
38 - 120
succinyl-Thr-Pro-Phe-4-nitroanilide
13 - 21
succinyl-Val-Pro-Leu-4-nitroanilide
1.2 - 8.7
succinyl-Val-Pro-Met-4-nitroanilide
57 - 75
succinyl-Val-Pro-Phe-4-nitroanilide
130 - 400
succinyl-Val-Pro-Pro-Phe-SCH2C6H5
5.6 - 8.4
succinyl-Val-Pro-Trp-4-nitroanilide
5.5 - 19
succinyl-Val-Pro-Tyr-4-nitroanilide
0.93
Ala-Ala-Pro-Leu-4-nitroanilide
wild type enzyme
3.9
Ala-Ala-Pro-Leu-4-nitroanilide
mutant enzyme A216G
19.3
Ala-Ala-Pro-Leu-4-nitroanilide
-
wild type enzyme
0.098
Ala-Ala-Pro-Met-4-nitroanilide
wild type enzyme
13
Ala-Ala-Pro-Met-4-nitroanilide
mutant enzyme A216G
23
Ala-Ala-Pro-Met-4-nitroanilide
-
wild type enzyme
0.028
Ala-Ala-Pro-Phe-4-nitroanilide
wild type enzyme
16
Ala-Ala-Pro-Phe-4-nitroanilide
mutant enzyme A216G
143
Ala-Ala-Pro-Phe-4-nitroanilide
-
wild type enzyme
65
angiotensin I
-
-
140
angiotensin I
-
glycosylated enzyme
143
angiotensin I
-
deglycosylated enzyme
24.7
Big endothelin-1
-
untreated enzyme
25.6
Big endothelin-1
-
deglycosylated enzyme
1.25
succinyl-Ala-Ala-Pro-Phe-4-nitroanilide
-
enzyme form 1E
1.66
succinyl-Ala-Ala-Pro-Phe-4-nitroanilide
-
enzyme form 1B
2.33
succinyl-Ala-Ala-Pro-Phe-4-nitroanilide
-
enzyme form 1A
2.54
succinyl-Ala-Ala-Pro-Phe-4-nitroanilide
-
enzyme form 1D
2.84
succinyl-Ala-Ala-Pro-Phe-4-nitroanilide
-
enzyme form 1C
17.5
succinyl-Ala-Ala-Pro-Phe-4-nitroanilide
-
pH 7.5, 22°C
65
succinyl-Ala-Ala-Pro-Phe-4-nitroanilide
-
-
38
succinyl-Ala-Pro-Phe-4-nitroanilide
-
-
51
succinyl-Ala-Pro-Phe-4-nitroanilide
-
-
86
succinyl-epsilon-(2-picolinyl)Lys-Val-Pro-Phe-4-nitroanilide
-
-
480
succinyl-epsilon-(2-picolinyl)Lys-Val-Pro-Phe-4-nitroanilide
-
-
56
succinyl-Gln-Pro-Phe-4-nitroanilide
-
-
86
succinyl-Gln-Pro-Phe-4-nitroanilide
-
-
9.2
succinyl-Glu-Pro-Phe-4-nitroanilide
-
-
61
succinyl-Glu-Pro-Phe-4-nitroanilide
-
-
53
succinyl-Glu-Val-Pro-Phe-4-nitroanilide
-
-
68
succinyl-Glu-Val-Pro-Phe-4-nitroanilide
-
-
2.5
succinyl-L-Ala-L-Ala-L-Pro-L-Phe-4-nitroanilide
-
in the presence of heparin, at pH 7.4 and 37°C
3.6
succinyl-L-Ala-L-Ala-L-Pro-L-Phe-4-nitroanilide
-
in the absence of heparin, at pH 7.4 and 37°C
12.6
succinyl-L-Ala-L-Ala-L-Pro-L-Phe-thiobenzyl ester
-
in the absence of heparin, at pH 7.4 and 37°C
17.8
succinyl-L-Ala-L-Ala-L-Pro-L-Phe-thiobenzyl ester
-
in the presence of heparin, at pH 7.4 and 37°C
37
succinyl-Leu-Pro-Phe-4-nitroanilide
-
-
77
succinyl-Leu-Pro-Phe-4-nitroanilide
-
-
19
succinyl-Leu-Val-Pro-Phe-4-nitroanilide
-
-
79
succinyl-Leu-Val-Pro-Phe-4-nitroanilide
-
-
14
succinyl-Lys-Pro-Phe-4-nitroanilide
-
-
32
succinyl-Lys-Pro-Phe-4-nitroanilide
-
-
58
succinyl-Lys-Val-Pro-Phe-4-nitroanilide
-
-
66
succinyl-Lys-Val-Pro-Phe-4-nitroanilide
-
-
25
succinyl-Met-Pro-Phe-4-nitroanilide
-
-
100
succinyl-Met-Pro-Phe-4-nitroanilide
-
-
25
succinyl-Met-Val-Pro-Phe-4-nitroanilide
-
-
30
succinyl-Met-Val-Pro-Phe-4-nitroanilide
-
-
53
succinyl-Met-Val-Pro-Phe-4-nitroanilide
-
-
7.1
succinyl-Phe-Ala-Phe-4-nitroanilide
-
-
10
succinyl-Phe-Ala-Phe-4-nitroanilide
-
-
3.9
succinyl-Phe-Gln-Phe-4-nitroanilide
-
-
25
succinyl-Phe-Gln-Phe-4-nitroanilide
-
-
0.9
succinyl-Phe-Glu-Phe-4-nitroanilide
-
-
8.4
succinyl-Phe-Glu-Phe-4-nitroanilide
-
-
7.5
succinyl-Phe-Leu-Phe-4-nitroanilide
-
-
17
succinyl-Phe-Leu-Phe-4-nitroanilide
-
-
19
succinyl-Phe-Leu-Phe-4-nitroanilide
-
-
5.9
succinyl-Phe-Met-Phe-4-nitroanilide
-
-
8.2
succinyl-Phe-Met-Phe-4-nitroanilide
-
-
17
succinyl-Phe-Pro-Phe-4-nitroanilide
-
-
24
succinyl-Phe-Pro-Phe-4-nitroanilide
-
-
28
succinyl-Phe-Pro-Phe-4-nitroanilide
-
-
11
succinyl-Phe-Pro-Thr-Phe-4-nitroanilide
-
-
19
succinyl-Phe-Pro-Thr-Phe-4-nitroanilide
-
-
5.4
succinyl-Phe-Ser-Phe-4-nitroanilide
-
-
6.2
succinyl-Phe-Ser-Phe-4-nitroanilide
-
-
9.3
succinyl-Phe-Thr-Phe-4-nitroanilide
-
-
10
succinyl-Phe-Thr-Phe-4-nitroanilide
-
-
4
succinyl-Phe-Val-Phe-4-nitroanilide
-
-
15
succinyl-Phe-Val-Phe-4-nitroanilide
-
-
24
succinyl-Phe-Val-Pro-Phe-4-nitroanilide
-
-
33
succinyl-Phe-Val-Pro-Phe-4-nitroanilide
-
-
56
succinyl-Phe-Val-Pro-Phe-4-nitroanilide
-
-
20
succinyl-Ser-Pro-Phe-4-nitroanilide
-
-
38
succinyl-Ser-Pro-Phe-4-nitroanilide
-
-
38
succinyl-Thr-Pro-Phe-4-nitroanilide
-
-
65
succinyl-Thr-Pro-Phe-4-nitroanilide
-
-
120
succinyl-Thr-Pro-Phe-4-nitroanilide
-
-
13
succinyl-Val-Pro-Leu-4-nitroanilide
-
-
21
succinyl-Val-Pro-Leu-4-nitroanilide
-
-
1.2
succinyl-Val-Pro-Met-4-nitroanilide
-
-
5
succinyl-Val-Pro-Met-4-nitroanilide
-
-
8.7
succinyl-Val-Pro-Met-4-nitroanilide
-
-
57
succinyl-Val-Pro-Phe-4-nitroanilide
-
-
75
succinyl-Val-Pro-Phe-4-nitroanilide
-
-
130
succinyl-Val-Pro-Pro-Phe-SCH2C6H5
-
-
400
succinyl-Val-Pro-Pro-Phe-SCH2C6H5
-
-
5.6
succinyl-Val-Pro-Trp-4-nitroanilide
-
-
8.4
succinyl-Val-Pro-Trp-4-nitroanilide
-
-
5.5
succinyl-Val-Pro-Tyr-4-nitroanilide
-
-
19
succinyl-Val-Pro-Tyr-4-nitroanilide
-
-