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3.4.21.35: tissue kallikrein

This is an abbreviated version!
For detailed information about tissue kallikrein, go to the full flat file.

Word Map on EC 3.4.21.35

Reaction

Preferential cleavage of Arg-/- bonds in small molecule substrates. Highly selective action to release kallidin (lysyl-bradykinin) from kininogen involves hydrolysis of Met-/- or Leu-/-. The rat enzyme is unusual in liberating bradykinin directly from autologous kininogens by cleavage at two Arg-/- bonds =

Synonyms

bradykininogenase, callicrein, depot-Padutin, dilminal D, EC 3.4.21.8, EC 3.4.4.21, EMSP1, GK1, glandular kallikrein, glandular kallikrein 2, glandular kallikrein 24, glandular kallikrein-2, glumorin, HK1, hK10, hK11, hK13, hK14, hK3, hK5, hK6, hK8, HSCTE, HUK, K1, K2, Kailikang, Kal, kallidinogenase, kallikrein, kallikrein 1, kallikrein 24, kallikrein-related peptidase, kallikrein-related peptidase 10, kallikrein-related peptidase 2, kallikrein-related peptidase 7, kidney/pancreas/salivary gland kallikrein, kininogenase, kininogenin, KLK, KLK-L1 protein, KLK-L2 protein, KLK-L3, KLK-S3, KLK1, KLK10, KLK11, KLK15, KLK2, KLK3, KLK4, KLK5, KLK6, KLK7, KLK9, mK1, mK13, mK22, mK24, mK9, More, neurosin, onokrein P., P1 kallikrein, padreatin, padutin, pancreatic kallikrein, pancreatic/renal kallikrein, PPK, Prk, pro-renin-converting enzyme, prokallikrein, prostase, prostase/KLK-L1/ARM1/PRSS17, prostate specific antigen, protease M, PS kallikrein, PSA, PSA/KLK3, renal kallikrein, renal tissue kallikrein, RSGK-50, RUK, S01.160, S1 kallikrein, S2 kallikrein, S3 kallikrein, salivary kallikrein, SEV, skeletal muscle kallikrein, submandibular enzymatic vasoconstrictor, T-kininogenase, tissue kallidinogenase, tissue kallikrein, tissue kallikrein 1, tissue kallikrein 11, tissue kallikrein 15, tissue kallikrein 4, tissue kallikrein 9, TK, trypsin-like serine protease, UKLK, urinary kallidinogenase, urinary kallikrein, urinary tissue kallikrein, urokallikrein, zyme

ECTree

     3 Hydrolases
         3.4 Acting on peptide bonds (peptidases)
             3.4.21 Serine endopeptidases
                3.4.21.35 tissue kallikrein

KCat KM Value

KCat KM Value on EC 3.4.21.35 - tissue kallikrein

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kcat/KM VALUE [1/mMs-1]
SUBSTRATE
ORGANISM
UNIPROT
COMMENTARY hide
LITERATURE
IMAGE
22
Abz-ALFSSKQ-EDDnp
-
at pH 7.5 and 37°C
27
Abz-FLFSSKQ-EDDnp
-
at pH 7.5 and 37°C
1067
Abz-FRSSR-Q-EDDnp
pH and temperature not specified in the publication
12780
Abz-GFSPFRSLRI-Q-EDDnp
pH and temperature not specified in the publication
88500
Abz-GFSPFRSSRI-Q-EDDnp
pH and temperature not specified in the publication
5
Abz-GLFSSKQ-EDDnp
-
at pH 7.5 and 37°C
30
Abz-HLFSSKQ-EDDnp
-
at pH 7.5 and 37°C
21
Abz-ILFSSKQ-EDDnp
-
at pH 7.5 and 37°C
6.3
Abz-KAFSSKQ-EDDnp
-
at pH 7.5 and 37°C
5.7
Abz-KFFSSKQ-EDDnp
-
at pH 7.5 and 37°C
25
Abz-KLFFSK-EDDnp
-
at pH 7.5 and 37°C
47
Abz-KLFRSK-EDDnp
-
at pH 7.5 and 37°C
69
Abz-KLFSAKQ-EDDnp
-
at pH 7.5 and 37°C
15
Abz-KLFSGKQ-EDDnp
-
at pH 7.5 and 37°C
31
Abz-KLFSIKQ-EDDnp
-
at pH 7.5 and 37°C
41
Abz-KLFSLKQ-EDDnp
-
at pH 7.5 and 37°C
16
Abz-KLFSNKQ-EDDnp
-
at pH 7.5 and 37°C
100
Abz-KLFSRKQ-EDDnp
-
at pH 7.5 and 37°C
16
Abz-KLFSSDQ-EDDnp
-
at pH 7.5 and 37°C
39
Abz-KLFSSEQ-EDDnp
-
at pH 7.5 and 37°C
53
Abz-KLFSSGQ-EDDnp
-
at pH 7.5 and 37°C
6
Abz-KLFSSIQ-EDDnp
-
at pH 7.5 and 37°C
55
Abz-KLFSSK-EDDnp
-
at pH 7.5 and 37°C
55
Abz-KLFSSKQ-EDDnp
-
at pH 7.5 and 37°C
25
Abz-KLFSSLQ-EDDnp
-
at pH 7.5 and 37°C
16
Abz-KLFSSNQ-EDDnp
-
at pH 7.5 and 37°C
33
Abz-KLFSSQQ-EDDnp
-
at pH 7.5 and 37°C
106
Abz-KLFSSRQ-EDDnp
-
at pH 7.5 and 37°C
73
Abz-KLFSSSQ-EDDnp
-
at pH 7.5 and 37°C
6
Abz-KLFSSVQ-EDDnp
-
at pH 7.5 and 37°C
130
Abz-KLFSVKQ-EDDnp
-
at pH 7.5 and 37°C
15
Abz-KLFTSK-EDDnp
-
at pH 7.5 and 37°C
17
Abz-KLFWSK-EDDnp
-
at pH 7.5 and 37°C
250
Abz-KLYSSK-EDDnp
-
at pH 7.5 and 37°C
6.4
Abz-KPFSSKQ-EDDnp
-
at pH 7.5 and 37°C
20
Abz-KVFSSKQ-EDDnp
-
at pH 7.5 and 37°C
6
Abz-KYFSSKQ-EDDnp
-
at pH 7.5 and 37°C
15
Abz-LLFSSKQ-EDDnp
-
at pH 7.5 and 37°C
2
Abz-MISLMKLP-Q-EDDnp
pH and temperature not specified in the publication
471
Abz-MISLMKRP-Q-EDDnp
pH and temperature not specified in the publication
165
Abz-NLFSSKQ-EDDnp
-
at pH 7.5 and 37°C
29
Abz-QLFSSKQ-EDDnp
-
at pH 7.5 and 37°C
32
Abz-RLFSSKQ-EDDnp
-
at pH 7.5 and 37°C
62
Abz-VLFSSKQ-EDDnp
-
at pH 7.5 and 37°C